Address https://gelex.eu/eli/EU/regulation/2007/129@2007-02-12/en

Contents

1. Preamble
2. 1. Article 1
   2. Article 2
   3. Article 3
   4. Article 4
   5. Article 5
   6. Article 6
3. ANNEX
4. ANNEX I List of international non-proprietary names (INNs) to be added to the list of products receiving duty-free treatment included in Annex 3 to Commission Regulation (EC) No 1549/2006
5. ANNEX II List of prefixes and suffixes which, in combination with the INNs of Annex 3 to Regulation (EC) No 1549/2006, describe the salts, esters or hydrates of INNs; these salts, esters and hydrates are free of duty, on condition that they are classifiable in the same six-digit HS-subheading as the corresponding INN
6. ANNEX III List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be added to the list of products receiving duty-free treatment included in Annex 6 to Regulation (EC) No 1549/2006
7. ANNEX IV List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be withdrawn from the list of products receiving duty-free treatment included in Annex 6 to Regulation (EC) No 1549/2006

THE COUNCIL OF THE EUROPEAN UNION,

Having regard to the Treaty establishing the European Community, and in particular Article 133 thereof,

Having regard to the proposal from the Commission,

Whereas:

(1) In the course of the Uruguay Round negotiations, the Community and a number of countries agreed that duty-free treatment should be granted to pharmaceutical products falling within the Harmonised System (HS) Chapter 30 and HS headings 2936, 2937, 2939 and 2941 as well as to designated pharmaceutical active ingredients bearing an international non-proprietary name (INN) from the World Health Organisation, specified salts, esters or hydrates of such INNs, and designated intermediates used for the production and manufacture of finished products.

(2) The results of the discussions, as set out in the record of discussions, were incorporated into the tariff schedules of the participants, annexed to the Marrakesh Protocol to the GATT 1994.

(3) Participants concluded that representatives of the WTO members, party to the record of discussions, would meet under the auspices of the WTO Council for Trade in Goods, normally at least once every three years to review the product coverage with a view to including, by consensus, additional pharmaceutical products for tariff elimination.

(4) In the course of three such reviews it was concluded that a certain number of additional INNs and intermediates used for production and manufacture of finished pharmaceuticals should be granted duty-free treatment, that certain of these intermediates should be transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs should be expanded.

(5) Council Regulation (EEC) No 2658/87 of 23 July 1987 on the tariff and statistical nomenclature and on the Common Customs Tariff established the Combined Nomenclature (CN) and set out the conventional duty rates of the Common Customs Tariff.

(6) Regulation (EEC) No 2658/87 should therefore be amended accordingly,

HAS ADOPTED THIS REGULATION:

Article 1

As from 1 January 2007 the Community shall extend duty-free treatment to the INNs listed in Annex I.

Article 2

As from 1 January 2007 the list of prefixes and suffixes which, in combination with the INNs, describe the salts, esters or hydrates of INNs which are also eligible for duty-free treatment, on condition that they are classifiable in the same six-digit HS-subheading as the corresponding INN, shall be replaced by the list in Annex II.

Article 3

As from 1 January 2007 the Community shall extend duty-free treatment to the intermediates used in the production and manufacture of pharmaceutical products listed in Annex III.

Article 4

As from 1 January 2007 the intermediates listed in Annex IV shall no longer benefit from duty-free treatment.

Article 5

Annexes 3, 4 and 6 of Section II of Part three of Annex I to Regulation (EEC) No 2658/87 (Lists of pharmaceutical substances which qualify for duty-free treatment) shall be amended accordingly.

Article 6

This Regulation shall enter into force on the day following its publication in the Official Journal of the European Union.

This Regulation shall be binding in its entirety and directly applicable in all Member States. Done at Brussels, 12 February 2007. For the Council The President F.-W. Steinmeier

ANNEX

ANNEX I List of international non-proprietary names (INNs) to be added to the list of products receiving duty-free treatment included in Annex 3 to Commission Regulation (EC) No 1549/2006

ID No CN code CAS RN Name 696 28429080 12539-23-0 vangatalcite 572 28439090 129580-63-8 satraplatin 413 28439090 141977-79-9 miriplatin 223 28439090 146665-77-2 eptaplatin 682 28439090 172903-00-3 triplatin tetranitrate 504 28439090 181630-15-9 picoplatin 807 28439090 274679-00-4 padoporfin 629 28444030 131608-78-1 technetium (99mTc) nitridocade 628 28444030 225239-31-6 technetium (99mTc) fanolesomab 711 28444030 476413-07-7 yttrium (90Y) tacatuzumab tetraxetan (yttrium (90Y) tacatuzumab) 738 28459010 474641-19-5 deutolperisone 283 28469000 193901-90-5 gadofosveset 284 28469000 227622-74-4 gadomelitol 281 28469000 280776-87-6 gadocoletic acid 282 28469000 544697-52-1 gadodenterate 761 29033990 354-92-7 perflisobutane 497 29033990 355-25-9 perflubutane 495 29033990 355-42-0 perflexane 498 29033990 76-19-7 perflutren 496 29034700 307-43-7 perflubrodec 328 29061900 163217-09-2 inecalcitol 727 29061900 524067-21-8 becocalcidiol 21 29072900 57-91-0 alfatradiol 464 29094990 128607-22-7 ospemifene 66 29094990 302904-82-1 atocalcitol 270 29094990 341524-89-8 fispemifene 592 29095090 3380-30-1 soneclosan 335 29144090 158440-71-2 irofulven 803 29147000 274925-86-9 nebicapone 56 29159080 185517-21-9 arundic acid 87 29163900 153559-49-0 bexarotene 640 29181985 121009-77-6 tenivastatin 659 29181985 156965-06-9 tisocalcitate 750 29181985 54845-95-3 icomucret 677 29189990 157283-68-6 travoprost 744 29189990 161172-51-6 etalocib 294 29189990 183293-82-5 gemcabene 643 29189990 251565-85-2 tesaglitazar 757 29189990 476436-68-7 naveglitazar 436 29213099 219810-59-0 neramexane 153 29214980 186495-49-8 delucemine 124 29214980 226256-56-0 cinacalcet 367 29214980 33817-09-3 levmetamfetamine 234 29221980 119618-22-3 esoxybutynin 611 29221980 146376-58-1 talibegron 596 29221980 148717-90-2 squalamine 266 29221980 162359-55-9 fingolimod 683 29221980 186139-09-3 trodusquemine 193 29221980 190258-12-9 edronocaine 709 29221980 207916-33-4 xidecaflur 391 29221980 36144-08-8 mantabegron 644 29221980 98774-23-3 tesmilifene 626 29222900 148717-54-8 tecalcet 619 29222900 175591-23-8 tapentadol 440 29222900 90060-42-7 nolomirole 230 29223900 33643-46-8 esketamine 198 29224995 176199-48-7 eglumetad (eglumegad) 310 29224995 198022-65-0 icofungipen 386 29224995 220991-20-8 lumiracoxib 554 29224995 220991-32-2 robenacoxib 103 29225000 135306-78-4 caloxetic acid 72 29225000 187219-95-0 axomadol 278 29225000 193901-91-6 fosveset 589 29225000 252920-94-8 solabegron 551 29225000 255734-04-4 ritobegron 752 29225000 269079-62-1 isalmadol 261 29225000 286930-03-8 fesoterodine 238 29225000 37178-37-3 etilevodopa 399 29225000 7101-51-1 melevodopa 161 29225000 93413-62-8 desvenlafaxine 110 29241900 1188-38-1 carglumic acid 632 29241900 250694-07-6 teglicar 692 29241900 92262-58-3 valrocemide 603 29242995 112522-64-2 tacedinaline 36 29242995 119363-62-1 amiglumide 195 29242995 131179-95-8 efaproxiral 528 29242995 133865-88-0 ralfinamide 567 29242995 133865-89-1 safinamide 735 29242995 147497-64-1 davasaicin 71 29242995 156740-57-7 axitirome 434 29242995 163000-63-3 neboglamine (nebostinel) 26 29242995 173334-57-1 aliskiren 347 29242995 175481-36-4 lacosamide (erlosamide) 332 29242995 181872-90-2 iosimenol 568 29242995 183990-46-7 salcaprozic acid 279 29242995 188196-22-7 frakefamide 601 29242995 193079-69-5 tabimorelin 462 29242995 196618-13-0 oseltamivir 349 29242995 209394-27-4 ladostigil 828 29242995 220847-86-9 valategrast 614 29242995 228266-40-8 taltobulin 668 29242995 260980-89-0 topilutamide 720 29242995 387825-03-8 salclobuzic acid 772 29242995 441765-98-6 talaglumetad 51 29242995 67346-49-0 arformoterol 449 29252900 146510-36-3 olanexidine 45 29252900 170368-04-4 anisperimus 494 29252900 229614-55-5 peramivir 737 29252900 287096-87-1 delmitide 35 29252900 346735-24-8 amelubant 642 29269095 108605-62-5 teriflunomide 121 29269095 153259-65-5 cilomilast 801 29269095 202057-76-9 manitimus 428 29269095 220641-11-2 naminidil 219 29280090 130579-75-8 eplivanserin 570 29280090 149400-88-4 sardomozide 777 29280090 154039-60-8 marimastat 798 29280090 203737-93-3 istaroxime 576 29280090 352513-83-8 semapimod 398 29280090 76144-81-5 meldonium 75 29299000 136470-65-0 banoxantrone 69 29299000 166518-60-1 avasimibe 172 29299000 168021-79-2 disufenton sodium 833 29309030 583-91-5 desmeninol 233 29309085 101973-77-7 esonarimod 53 29309085 112111-43-0 armodafinil 731 29309085 158382-37-7 canfosfamide 618 29309085 179545-77-8 tanomastat 766 29309085 187870-78-6 rimeporide 196 29309085 202340-45-2 eflucimibe 165 29309085 29335-92-0 dextiopronin 760 29309085 496050-39-6 pemaglitazar 250 29309085 59973-80-7 exisulind 307 29310095 133208-93-2 ibrolipim 372 29310095 63132-38-7 lidadronic acid 556 29321900 156722-18-8 rostafuroxin 410 29321900 393101-41-2 milataxel 58 29322985 109791-32-4 ascorbyl gamolenate 171 29322985 127943-53-7 disermolide 272 29322985 140616-46-2 fluorescein lisicol 19 29322985 150785-53-8 alemcinal 416 29322985 154738-42-8 mitemcinal 38 29322985 161262-29-9 amotosalen 555 29322985 162011-90-7 rofecoxib 574 29322985 165108-07-6 selamectin 269 29322985 189954-96-9 firocoxib 469 29329950 186040-50-6 paclitaxel ceribate 273 29329970 114870-03-0 fondaparinux sodium 229 29329970 128196-01-0 escitalopram 463 29329970 137275-81-1 osemozotan 312 29329970 149920-56-9 idraparinux sodium 211 29329970 167256-08-8 enrasentan 150 29329970 171092-39-0 defoslimod 650 29329970 175013-73-7 tidembersat 455 29329970 181296-84-4 omigapil 743 29329970 185955-34-4 eritoran 461 29329970 186348-23-2 ortataxel 529 29329970 196597-26-9 ramelteon 467 29329970 280585-34-4 oxeglitazar 375 29329970 329306-27-6 lirimilast 163 29329970 51372-29-3 dexbudesonide 54 29329970 75887-54-6 artemotil 314 29329970 81267-65-4 idronoxil 667 29329985 175013-84-0 tonabersat 109 29329985 184653-84-7 carabersat 55 29329985 81496-81-3 artenimol 769 29329990 343306-71-8 sugammadex 224 29332990 129805-33-0 eptotermin alfa 255 29332990 134183-95-2 fampronil 249 29332990 141758-74-9 exenatide 806 29332990 144689-24-7 olmesartan 176 29332990 149838-23-3 doranidazole 268 29332990 150586-58-6 fipamezole 578 29332990 154906-40-8 semparatide 204 29332990 159075-60-2 emfilermin 209 29332990 159519-65-0 enfuvirtide 472 29332990 162394-19-6 palifermin 89 29332990 163796-60-9 bifarcept 321 29332990 170105-16-5 imidafenacin 657 29332990 178823-49-9 tiplimotide 253 29332990 189353-31-9 fadolmidine (radolmidine) 389 29332990 200074-80-2 lusupultide 126 29332990 213027-19-1 cipralisant 541 29332990 219527-63-6 repifermin 605 29332990 220712-29-8 tadekinig alfa 167 29332990 246539-15-1 dibotermin alfa 536 29332990 259188-38-0 rebimastat 790 29332990 444069-80-1 dapiclermine 396 29332990 478166-15-3 mecasermin rinfabate 134 29333999 0-00-0 crobenetine 591 29333999 0-00-0 solimastat 159 29333999 100643-71-8 desloratadine 299 29333999 103766-25-2 gimeracil 342 29333999 112568-12-4 iturelix 637 29333999 113712-98-4 tenatoprazole 232 29333999 119141-88-7 esomeprazole 804 29333999 119229-65-1 nerispirdine 308 29333999 119515-38-7 icaridin 29 29333999 120241-31-8 alvameline 411 29333999 128420-61-1 minopafant 678 29333999 134234-12-1 traxoprodil 519 29333999 134457-28-6 prazarelix 791 29333999 138530-94-6 dexlansoprazole 800 29333999 138530-95-7 levolansoprazole 712 29333999 142852-50-4 zanapezil 252 29333999 147116-64-1 ezlopitant 394 29333999 147116-67-4 maropitant 180 29333999 150337-94-3 ecalcidene 350 29333999 153322-05-5 lanicemine 815 29333999 15585-43-0 rivanicline 30 29333999 156053-89-3 alvimopan 333 29333999 166181-63-1 ipravacaine 707 29333999 168266-90-8 vofopitant 549 29333999 168273-06-1 rimonabant 215 29333999 170364-57-5 enzastaurin 318 29333999 172152-36-2 ilaprazole 107 29333999 178979-85-6 capravirine 655 29333999 179033-51-3 timcodar 262 29333999 183305-24-0 fidexaban 809 29333999 188396-77-2 paliroden 158 29333999 188913-58-8 dersalazine 125 29333999 190648-49-8 cipemastat 465 29333999 193153-04-7 otamixaban 380 29333999 193275-84-2 lonafarnib 645 29333999 195875-84-4 tesofensine 623 29333999 198283-73-7 tebanicline 507 29333999 198480-55-6 pipendoxifene 65 29333999 198904-31-3 atazanavir 199 29333999 198958-88-2 elarofiban 341 29333999 201605-51-8 itriglumide 91 29333999 202189-78-4 bilastine 240 29333999 202409-33-4 etoricoxib 649 29333999 202590-69-0 ticalopride 325 29333999 204205-90-3 indibulin 136 29333999 211914-51-1 dabigatran 137 29333999 211915-06-9 dabigatran etexilate 701 29333999 212141-54-3 vatalanib 74 29333999 215529-47-8 bamirastine 10 29333999 227940-00-3 adekalant 699 29333999 249296-44-4 varenicline 797 29333999 252870-53-4 ispronicline 76 29333999 263562-28-3 barixibat 594 29333999 284461-73-0 sorafenib 821 29333999 288104-79-0 surinabant 52 29333999 289893-25-0 arimoclomol 721 29333999 370893-06-4 ancriviroc 392 29333999 376348-65-1 maraviroc 164 29333999 40431-64-9 dexmethylphenidate 316 29333999 58754-46-4 iferanserin 788 29333999 64881-21-6 caricotamide 409 29333999 72599-27-0 miglustat 627 29333999 75970-99-9 tecastemizole 579 29333999 98326-32-0 senazodan 448 29334910 167887-97-0 olamufloxacin 606 29334990 106635-80-7 tafenoquine 714 29334990 139233-53-7 zelandopam 25 29334990 144506-11-6 alilusem 397 29334990 146362-70-1 meclinertant (reminertant) 508 29334990 147511-69-1 pitavastatin (itavastatin) 506 29334990 149759-26-2 pinokalant 613 29334990 174636-32-9 talnetant 290 29334990 194804-75-6 garenoxacin 515 29334990 195532-12-8 pradofloxacin 352 29334990 197509-46-9 laniquidar 622 29334990 206873-63-4 tariquidar 288 29334990 213998-46-0 gantacurium chloride 717 29334990 241800-98-6 zoniporide 590 29334990 242478-37-1 solifenacin 492 29334990 257933-82-7 pelitinib 672 29334990 262352-17-0 torcetrapib 476 29334990 540769-28-6 palosuran 586 29334990 57695-04-2 sitamaquine 264 29335995 0-00-0 figopitant 660 29335995 103024-93-7 tiviciclovir 406 29335995 117414-74-1 midafotel 452 29335995 124265-89-0 omaciclovir 173 29335995 129716-58-1 dofequidar 102 29335995 133804-44-1 caldaret 366 29335995 138117-50-7 leteprinim 213 29335995 142217-69-4 entecavir 763 29335995 146464-95-1 pralatrexate 641 29335995 147127-20-6 tenofovir 531 29335995 147254-64-6 ranirestat 205 29335995 149950-60-7 emivirine 320 29335995 152459-95-5 imatinib 511 29335995 153537-73-6 plevitrexed 100 29335995 153808-85-6 cadrofloxacin 503 29335995 154889-68-6 pibrozelesin 718 29335995 167354-41-8 zosuquidar 174 29335995 170912-52-4 donitriptan 146 29335995 171714-84-4 darusentan 32 29335995 177036-94-1 ambrisentan 226 29335995 183321-74-6 erlotinib 768 29335995 186692-46-6 seliciclib 17 29335995 187949-02-6 albaconazole 381 29335995 192725-17-0 lopinavir 16 29335995 193681-12-8 alamifovir 691 29335995 195157-34-7 valomaciclovir 254 29335995 196612-93-8 falnidamol 547 29335995 199463-33-7 revaprazan 260 29335995 204267-33-4 feloprentan 450 29335995 204697-65-4 olcegepant 746 29335995 209799-67-7 forodesine 716 29335995 210245-80-0 zonampanel 162 29335995 220984-26-9 detiviciclovir 142 29335995 244767-67-7 dapivirine 208 29335995 259525-01-4 enecadin 241 29335995 269055-15-4 etravirine 439 29335995 290297-26-6 netupitant 566 29335995 324758-66-9 sabiporide 724 29335995 330784-47-9 avanafil 703 29335995 334476-46-9 vestipitant 753 29335995 336113-53-2 ispinesib 695 29335995 338992-00-0 vandetanib 725 29335995 354813-19-7 balicatib 616 29335995 387867-13-2 tandutinib 242 29335995 402595-29-3 etriciguat 522 29335995 443144-26-1 pruvanserin 548 29335995 500287-72-9 rilpivirine 147 29335995 569351-91-3 dasantafil 795 29335995 61337-87-9 esmirtazapine 222 29336980 179756-85-5 eptapirone 728 29336980 187393-00-6 bemotrizinol 512 29336980 69004-04-2 ponazuril 466 29336980 937-13-3 oteracil 235 29337900 138729-47-2 eszopiclone 354 29337900 142139-60-4 lapisteride 111 29337900 147568-66-9 carmoterol 88 29337900 148905-78-6 bexlosteride 296 29337900 160135-92-2 gemopatrilat 156 29337900 161982-62-3 depreotide 251 29337900 163222-33-1 ezetimibe 140 29337900 182821-27-8 daglutril 271 29337900 187523-35-9 flindokalner 120 29337900 188968-51-6 cilengitide 362 29337900 191732-72-6 lenalidomide 656 29337900 192185-72-1 tipifarnib 577 29337900 194413-58-6 semaxanib 355 29337900 248281-84-7 laquinimod 823 29337900 254964-60-8 tasquinimod 324 29337900 312753-06-3 indacaterol 787 29337900 357336-20-0 brivaracetam 818 29337900 357336-74-4 seletracetam 781 29337900 503612-47-3 apixaban 820 29337900 557795-19-4 sunitinib 231 29339930 104746-04-5 eslicarbazepine 181 29339930 112108-01-7 ecopipam 422 29339930 137975-06-5 mozavaptan 665 29339930 150683-30-0 tolvaptan 131 29339930 210101-16-9 conivaptan 370 29339930 29331-92-8 licarbazepine 500 29339940 144912-63-0 perzinfotel 378 29339940 168079-32-1 lixivaptan 423 29339940 174391-92-5 mozenavir 166 29339940 82059-50-5 dextofisopam 730 29339990 103597-45-1 bisoctrizole 597 29339990 106344-20-1 stannsoporfin 811 29339990 110078-46-1 plerixafor 610 29339990 110230-98-3 talaporfin 46 29339990 114560-48-4 apaziquone 778 29339990 129497-78-5 verteporfin 510 29339990 144510-96-3 pixantrone 544 29339990 144875-48-9 resiquimod 631 29339990 145158-71-0 tegaserod 588 29339990 149606-27-9 soblidotin 770 29339990 149682-77-9 talabostat 101 29339990 151878-23-8 calcobutrol 518 29339990 153804-05-8 pratosartan 758 29339990 154082-13-0 omocianine 442 29339990 156090-17-4 nortopixantrone 669 29339990 156090-18-5 topixantrone 371 29339990 156897-06-2 licofelone 267 29339990 160146-17-8 finrozole 582 29339990 160970-54-7 silodosin 311 29339990 169543-49-1 icrocaptide 700 29339990 172732-68-2 varespladib 435 29339990 173240-15-8 nemifitide 210 29339990 176644-21-6 eniporide 323 29339990 177469-96-4 implitapide 457 29339990 178040-94-3 opaviraline 28 29339990 179120-92-4 altinicline 97 29339990 179324-69-7 bortezomib 600 29339990 179386-43-7 sumanirole 357 29339990 180916-16-9 lasofoxifene 64 29339990 182316-31-0 ataquimast 329 29339990 186392-65-4 ingliforib 80 29339990 188696-80-2 becampanel 471 29339990 189198-30-9 pactimibe 421 29339990 189752-49-6 motexafin 822 29339990 192658-64-3 tasidotin 710 29339990 192939-46-1 ximelagatran 108 29339990 193273-66-4 capromorelin 276 29339990 194798-83-9 fosfluconazole 79 29339990 198481-32-2 bazedoxifene 149 29339990 201530-41-8 deferasirox 98 29339990 203258-60-0 brostallicin 454 29339990 204248-78-2 omiganan 295 29339990 204519-64-2 gemifloxacin 523 29339990 207993-12-2 pumafentrine 361 29339990 215808-49-4 lemuteporfin 826 29339990 21919-05-1 tretazicar 831 29339990 219680-11-2 zabofloxacin 526 29339990 244081-42-3 rafabegron 755 29339990 248919-64-4 linaprazan 652 29339990 251562-00-2 tifuvirtide 595 29339990 261944-46-1 soraprazan 705 29339990 274901-16-5 vildagliptin 557 29339990 284041-10-7 rostaporfin 767 29339990 361442-04-8 saxagliptin 447 29339990 38101-59-6 oglufanide 133 29339990 38609-97-1 cridanimod 481 29339990 396091-73-9 pasireotide 139 29339990 404951-53-7 dacinostat 192 29339990 433922-67-9 edratide 170 29339990 481658-94-0 dirlotapide 723 29339990 533927-56-9 atilmotin 773 29339990 637328-69-9 tanogitran 681 29339990 72741-87-8 tridolgosir 754 29339990 82059-51-6 levotofisopam 419 29341000 130112-42-4 mivotilate 144 29341000 139226-28-1 darbufelone 259 29341000 144060-53-7 febuxostat 646 29341000 145739-56-6 tetomilast 438 29341000 161600-01-7 netoglitazone 534 29341000 182760-06-1 ravuconazole 6 29341000 185106-16-5 acotiamide 553 29341000 185428-18-6 rivoglitazone 73 29341000 199113-98-9 balaglitazone 186 29341000 213411-83-7 edaglitazone 736 29341000 239101-33-8 deferitrin 122 29341000 300832-84-2 ciluprevir 15 29341000 341028-37-3 alagebrium chloride 819 29341000 342026-92-0 sipoglitazar 550 29341000 79714-31-1 risarestat 580 29342080 154189-40-9 sibenadet 344 29342080 176975-26-1 izonsteride 373 29342080 245116-90-9 lidorestat 387 29342080 367514-87-2 lurasidone 105 29349990 0-00-0 cangrelor 287 29349990 0-00-0 ganstigmine 509 29349990 0-00-0 pitrakinra 575 29349990 110299-05-3 selodenoson 365 29349990 111358-88-4 lestaurtinib 686 29349990 112984-60-8 ulifloxacin 676 29349990 114899-77-3 trabectedin 351 29349990 117276-75-2 lanimostim 776 29349990 120313-91-9 thrombomodulin alfa 408 29349990 120685-11-2 midostaurin 337 29349990 122970-40-5 isatoribine 129 29349990 123318-82-1 clofarabine 437 29349990 124584-08-3 nesiritide 647 29349990 130306-02-4 tezacitabine 390 29349990 135306-39-7 manifaxine 130 29349990 135463-81-9 coluracetam 505 29349990 137071-32-0 pimecrolimus 446 29349990 137215-12-4 odiparcil 812 29349990 137219-37-5 plitidepsin 207 29349990 143491-57-0 emtricitabine 95 29349990 144348-08-3 binodenoson 474 29349990 144598-75-4 paliperidone 451 29349990 144689-63-4 olmesartan medoxomil (olmesartan) 33 29349990 145514-04-1 amdoxovir 684 29349990 145918-75-8 troxacitabine 31 29349990 146426-40-6 alvocidib 585 29349990 147817-50-3 siramesine 569 29349990 148430-28-8 sarakalim 517 29349990 150322-43-3 prasugrel 49 29349990 151879-73-1 aprinocarsen 688 29349990 152735-23-4 upidosin 502 29349990 152811-62-6 piboserod 524 29349990 153062-94-3 pumosetrag 206 29349990 155030-63-0 emodepside 245 29349990 159351-69-6 everolimus 382 29349990 161178-07-0 lubazodone 256 29349990 161605-73-8 fanapanel 609 29349990 161832-65-1 talampanel 775 29349990 162635-04-3 temsirolimus 704 29349990 163521-12-8 vilazodone 3 29349990 167362-48-3 abetimus 330 29349990 169148-63-4 insulin detemir 562 29349990 169939-94-0 ruboxistaurin 48 29349990 170729-80-3 aprepitant 538 29349990 170861-63-9 reglitazar 513 29349990 171228-49-2 posaconazole 604 29349990 171596-29-5 tadalafil 11 29349990 171752-56-0 adrogolide 190 29349990 174402-32-5 edotecarin 796 29349990 174638-15-4 fosfluridine tidoxil 393 29349990 176161-24-3 maribavir 417 29349990 179602-65-4 mitratapid 201 29349990 181785-84-2 elvucitabine 57 29349990 182133-25-1 arzoxifene 5 29349990 182167-02-8 acolbifene 762 29349990 182415-09-4 piclozotan 289 29349990 183547-57-1 gantofiban 1 29349990 183849-43-6 abaperidone 293 29349990 184475-35-2 gefitinib 24 29349990 185229-68-9 alicaforsen 663 29349990 185954-27-2 tofimilast 384 29349990 187164-19-8 luliconazole 368 29349990 188630-14-0 liatermin 473 29349990 189681-70-7 aplindore (palindore) 148 29349990 189940-24-7 daxalipram 443 29349990 190977-41-4 oblimersen 309 29349990 192314-93-5 iclaprim 525 29349990 192374-14-4 radafaxine 379 29349990 192441-08-0 lomeguatrib 516 29349990 192755-52-5 pralnacasan 364 29349990 193700-51-5 leridistim 68 29349990 195733-43-8 atrasentan 132 29349990 195962-23-3 corifollitropin alfa 258 29349990 196808-45-4 farglitazar 402 29349990 198821-22-6 merimepodib 456 29349990 199685-57-9 onercept 191 29349990 204318-14-9 edotreotide 625 29349990 204512-90-3 tecadenoson 671 29349990 204658-47-9 torapsel 634 29349990 205887-54-3 telbermin 458 29349990 206254-79-7 opebacan 334 29349990 206260-33-5 irampanel 280 29349990 208848-19-5 freselestat 263 29349990 208993-54-8 fiduxosin 265 29349990 209342-40-5 finafloxacin 154 29349990 211448-85-0 denufosol 745 29349990 211735-76-1 farampator 388 29349990 214548-46-6 lusaperidone 814 29349990 215174-50-8 rimacalib 535 29349990 218298-21-6 razaxaban 543 29349990 219846-31-8 radequinil (resequinil) 257 29349990 221241-63-0 fandosentan 527 29349990 222834-30-2 ragaglitazar 563 29349990 223537-30-2 rupintrivir 99 29349990 223661-25-4 bulaquine 353 29349990 231277-92-2 lapatinib 359 29349990 247207-64-3 leconotide 322 29349990 250601-04-8 imiglitazar 8 29349990 250710-65-7 adargileukin alfa 228 29349990 251303-04-5 ertiprotafib 514 29349990 252260-02-9 posizolid 722 29349990 255730-18-8 artemifone 338 29349990 257277-05-7 iseganan 104 29349990 267243-28-7 canertinib 336 29349990 276690-58-5 iroxanadine 651 29349990 279215-43-9 tifenazoxide 118 29349990 282526-98-1 cetilistat 77 29349990 285571-64-4 barusiban 175 29349990 285983-48-4 doramapimod 81 29349990 290296-68-3 befetupitant 792 29349990 292634-27-6 dianicline 615 29349990 304853-42-7 tanaproget 50 29349990 305391-49-5 ardenermin 771 29349990 308240-58-6 talactoferrin alfa 598 29349990 308831-61-0 sufugolix 537 29349990 313348-27-5 regadenoson 326 29349990 325715-02-4 indiplon 187 29349990 328538-04-1 edifoligide 741 29349990 329744-44-7 embeconazole 425 29349990 331741-94-7 muraglitazar 759 29349990 331744-64-0 peliglitazar 825 29349990 333754-36-2 tesetaxel 635 29349990 3424-98-4 telbivudine 90 29349990 350992-10-8 bifeprunox 571 29349990 351862-32-3 sarizotan 202 29349990 361343-19-3 elzasonan 424 29349990 366017-09-6 mubritinib 552 29349990 366789-02-8 rivaroxaban 694 29349990 380886-95-3 valtorcitabine 673 29349990 40093-94-5 torcitabine 662 29349990 41941-56-4 tocladesine 799 29349990 434283-16-6 lecozotan 493 29349990 446022-33-9 pelitrexol 339 29349990 457913-93-8 ismomultin alfa 793 29349990 460738-38-9 ecallantide 155 29349990 506433-25-6 depelestat 414 29349990 507453-82-9 mirococept 84 29349990 566906-50-1 beminafil 764 29349990 575458-75-2 radotermin 783 29349990 583057-48-1 arasertaconazole 169 29349990 59985-21-6 diquafosol 813 29349990 625095-60-5 pradefovir 829 29349990 640281-90-9 valopicitabine 60 29349990 65576-45-6 asenapine 431 29349990 84472-85-5 navuridine 559 29349990 99755-59-6 rotigotine 599 29350090 0-00-0 sulamserod 317 29350090 123663-49-0 iguratimod 542 29350090 144980-29-0 repinotan 539 29350090 150375-75-0 relcovaptan 127 29350090 158751-64-5 clamikalant 39 29350090 161814-49-9 amprenavir 824 29350090 165538-40-9 terutroban 327 29350090 165668-41-7 indisulam 157 29350090 169590-41-4 deracoxib 115 29350090 169590-42-5 celecoxib 593 29350090 170858-33-0 sonepiprazole 658 29350090 174484-41-4 tipranavir 654 29350090 180200-68-4 tilmacoxib 128 29350090 180384-56-9 clazosentan 648 29350090 180384-57-0 tezosentan 679 29350090 180918-68-7 trecetilide 690 29350090 181695-72-7 valdecoxib 587 29350090 184036-34-8 sitaxentan 817 29350090 185913-78-4 satavaptan 520 29350090 192329-42-3 prinomastat 78 29350090 195533-53-0 batabulin 479 29350090 198470-84-7 parecoxib 145 29350090 206361-99-1 darunavir 40 29350090 209733-45-9 anatibant 621 29350090 210538-44-6 taprizosin 189 29350090 210891-04-6 edonentan 138 29350090 219311-44-1 dabuzalgron 698 29350090 224785-90-4 vardenafil 275 29350090 226700-79-4 fosamprenavir 666 29350090 233254-24-5 tomeglovir 63 29350090 254877-67-3 ataciguat 123 29350090 265114-23-6 cimicoxib 540 29350090 266359-83-5 reparixin 827 29350090 268203-93-6 udenafil 782 29350090 287405-51-0 apratastat 558 29350090 287714-41-4 rosuvastatin 784 29350090 290815-26-8 avosentan 376 29350090 321915-31-5 litomeglovir 182 29350090 381683-92-7 ecopladib 739 29350090 381683-94-9 efipladib 433 29350090 403604-85-3 nebentan 27 29362100 5300-03-8 alitretinoin 178 29362990 54573-75-0 doxercalciferol 810 29371900 147859-97-0 peforelin 346 29371900 159768-75-9 labradimil 4 29371900 178535-93-8 abrineurin 404 29371900 186018-45-1 metreleptin 374 29371900 204656-20-2 liraglutide 331 29371900 207748-29-6 insulin glulisine 151 29371900 214766-78-6 degarelix 491 29371900 218620-50-9 pegvisomant 630 29371900 287714-30-1 teduglutide 478 29371900 345663-45-8 parathyroid hormone 719 29372200 0-00-0 zoticasone 239 29372200 199331-40-3 etiprednol dicloacetate 674 29372300 110072-15-6 tosagestin 573 29372300 7690-08-6 segesterone 687 29372900 159811-51-5 uliprisnil 61 29372900 199396-76-4 asoprisnil 62 29372900 222732-94-7 asoprisnil ecamate 441 29372900 53016-31-2 norelgestromin 43 29372900 7753-60-8 anecortave 183 29375000 136892-64-3 ecraprost 92 29375000 155206-00-1 bimatoprost 608 29375000 209860-87-7 tafluprost 816 29375000 256382-08-8 rivenprost 383 29375000 333963-40-9 lubiprostone 197 29375000 63266-93-3 eganoprost 680 29375000 81846-19-7 treprostinil 427 29391900 152657-84-6 nalfurafine 756 29391900 20290-10-2 morphine glucuronide 407 29395900 151159-23-8 midaxifylline 340 29395900 155270-99-8 istradefylline 432 29395900 166374-49-8 naxifylline 247 29399900 0-00-0 exatecan alideximer 246 29399900 171335-80-1 exatecan 484 29399900 203066-49-3 pegamotecan 12 29399900 215604-75-4 afeletecan 168 29399900 220997-97-7 diflomotecan 740 29399900 220998-10-7 elomotecan 83 29399900 256411-32-2 belotecan 298 29399900 292618-32-7 gimatecan 561 29399900 91421-42-0 rubitecan 607 29400000 179067-42-6 tafluposide 93 29400000 187269-40-5 bimosiamose 277 29400000 488-69-7 fosfructose 653 29413000 220620-09-7 tigecycline 313 29415000 110480-13-2 idremcinal 468 29419000 0-00-0 ozogamicin 244 29419000 109545-84-8 evernimicin 726 29419000 119673-08-4 becatecarin 113 29419000 140128-74-1 cefmatilen 285 29419000 140637-86-1 galarubicin 177 29419000 148016-81-3 doripenem 482 29419000 152044-54-7 patupilone 227 29419000 153832-46-3 ertapenem 624 29419000 161715-24-8 tebipenem pivoxil (tebipenem) 112 29419000 162808-62-0 caspofungin 44 29419000 166663-25-8 anidulafungin 348 29419000 171047-47-5 ladirubicin 460 29419000 171099-57-3 oritavancin 141 29419000 171500-79-1 dalbavancin 636 29419000 173838-31-8 telithromycin 602 29419000 193811-33-5 tacapenem 117 29419000 205110-48-1 cethromycin 732 29419000 209467-52-7 ceftobiprole 708 29419000 21102-49-8 volpristin 565 29419000 211100-13-9 sabarubicin 685 29419000 217500-96-4 tulathromycin A + 280755-12-6 tulath. B tulathromycin 343 29419000 219989-84-1 ixabepilone 546 29419000 224452-66-8 retapamulin 114 29419000 234096-34-5 cefovecin 405 29419000 235114-32-6 micafungin 358 29419000 371918-51-3 (component A3), 371918-44-4 (component A4) latidectin 633 29419000 372151-71-8 telavancin 733 29419000 376653-43-9 ceftobiprole medocaril 693 29419000 56124-62-0 valrubicin 41 30021091 0-00-0 anatumomab mafenatox 217 30021091 0-00-0 epitumomab 301 30021091 0-00-0 hemoglobin glutamer 715 30021091 0-00-0 ziralimumab 475 30021091 188039-54-5 palivizumab 430 30021091 189261-10-7 natalizumab 675 30021091 192391-48-3 tositumomab 702 30021091 195158-85-1 vepalimomab 412 30021091 195189-17-4 minretumomab 400 30021091 196078-29-2 mepolizumab 560 30021091 197099-66-4 rovelizumab 302 30021091 197462-97-8 hemoglobin raffimer 420 30021091 202833-07-6 morolimumab 67 30021091 202833-08-7 atorolimumab 119 30021091 205923-56-4 cetuximab 221 30021091 205923-57-5 epratuzumab 306 30021091 206181-63-7 ibritumomab tiuxetan 225 30021091 211323-03-4 erlizumab 459 30021091 213327-37-8 oregovomab 96 30021091 214559-60-1 bivatuzumab 194 30021091 214745-43-4 efalizumab 20 30021091 216503-57-0 alemtuzumab 418 30021091 216503-58-1 mitumomab 581 30021091 216669-97-5 sibrotuzumab 86 30021091 216974-75-3 bevacizumab 345 30021091 219649-07-7 labetuzumab 185 30021091 219685-50-4 eculizumab 501 30021091 219685-93-5 pexelizumab 706 30021091 219716-33-3 visilizumab 297 30021091 220578-59-6 gemtuzumab 564 30021091 220651-94-5 ruplizumab 620 30021091 235428-87-2 taplitumomab paptox 545 30021091 241473-69-8 reslizumab 453 30021091 242138-07-4 omalizumab 292 30021091 244096-20-6 gavilimomab 360 30021091 250242-54-7 lemalesomab 670 30021091 252662-47-8 toralizumab 218 30021091 263547-71-3 epitumomab cituxetan 47 30021091 267227-08-7 apolizumab 403 30021091 272780-74-2 metelimumab 363 30021091 285985-06-0 lerdelimumab 584 30021091 288392-69-8 siplizumab 184 30021091 292819-64-8 ecromeximab 639 30021091 299423-37-3 teneliximab 274 30021091 326859-36-3 fontolizumab 480 30021091 331243-22-2 pascolizumab 7 30021091 331731-18-1 adalimumab 697 30021091 336801-86-6 vapaliximab 477 30021091 339177-26-3 panitumumab 395 30021091 339186-68-4 matuzumab 530 30021091 347396-82-1 ranibizumab 82 30021091 356547-88-1 belimumab 286 30021091 357613-77-5 galiximab 385 30021091 357613-86-6 lumiliximab 85 30021091 375348-49-5 bertilimumab 661 30021091 375823-41-9 tocilizumab 612 30021091 380610-22-0 talizumab 499 30021091 380610-27-5 pertuzumab 59 30021091 395639-53-9 aselizumab 106 30021091 400010-39-1 cantuzumab mertansine 116 30021091 428863-50-7 certolizumab pegol 200 30021091 468715-71-1 elsilimomab 300 30021091 476181-74-5 golimumab 521 30021091 499212-74-7 pritumumab 689 30021091 502496-16-4 urtoxazumab 9 30021091 503605-66-1 adecatumumab 789 30021091 509077-98-9 catumaxomab 794 30021091 509077-99-0 ertumaxomab 774 30021091 521079-87-8 tefibazumab 729 30021091 537694-98-7 besilesomab 830 30021091 558480-40-3 volociximab 765 30021091 565451-13-0 raxibacumab 369 30021091 569658-79-3 libivirumab 248 30021091 569658-80-6 exbivirumab 808 30021091 595566-61-3 pagibaximab 751 30021091 635715-01-4 inotuzumab ozogamicin 785 30021091 648895-38-9 bapineuzumab 713 30021091 652153-01-0 zanolimumab 802 30021091 658052-09-6 mapatumumab 832 30021091 667901-13-5 zalutumumab 805 30021091 679818-59-8 ofatumumab 319 30021095 149824-15-7 ilodecakin 42 30021095 163545-26-4 ancestim 236 30021095 185243-69-0 etanercept 188 30021095 187348-17-0 edodekin alfa 94 30021095 207137-56-2 binetrakin 143 30021095 209810-58-2 darbepoetin alfa 18 30021095 222535-22-0 alefacept 415 30021095 244130-01-6 mirostipen 291 30021095 246861-96-1 garnocestim 220 30021095 261356-80-3 epoetin delta 2 30021095 332348-12-6 abatacept 617 30021095 465540-87-8 taneptacogin alfa 749 30021095 479198-61-3 iboctadekin 742 30021095 604802-70-2 epoetin zeta 786 30021095 706808-37-9 belatacept 179 30021095 98530-76-8 drotrecogin alfa (activated) 780 30021099 84720-88-7 antithrombin alfa 70 30029090 223577-45-5 aviscumine 734 30029090 372075-36-0 cintredekin besudotox 779 35040000 9009-65-8 protamine sulfate 243 35079090 0-00-0 eufauserase 13 35079090 104138-64-9 agalsidase alfa 14 35079090 104138-64-9 agalsidase beta 533 35079090 134774-45-1 rasburicase 429 35079090 136653-69-5 nasaruplase beta 160 35079090 145137-38-8 desmoteplase 34 35079090 151912-11-7 amediplase 638 35079090 191588-94-0 tenecteplase 532 35079090 196488-72-9 ranpirnase 216 35079090 208576-22-1 epafipase 356 35079090 210589-09-6 laronidase 22 35079090 259074-76-5 alfimeprase 23 35079090 420784-05-0 alglucosidase alfa 315 35079090 50936-59-9 idursulfase (idusulfase) 747 35079090 552858-79-4 galsulfase 748 35079090 9074-87-7 glucarpidase 426 39069090 246527-99-1 mureletecan 485 39072021 0-00-0 pegaptanib 483 39072021 187139-68-0 pegacaristim 487 39072021 198153-51-4 peginterferon alfa-2a 489 39072021 204565-76-4 pegnartograstim 486 39072021 208265-92-3 pegfilgrastim 488 39072021 215647-85-1 peginterferon alfa-2b 490 39072021 330988-75-5 pegsunercept 470 39089000 263351-82-2 paclitaxel poliglumex 664 39119099 28210-41-5 tolevamer 377 39139000 329306-27-6 livaraparin calcium 152 39139000 9041-08-1 deligoparin sodium

ANNEX II List of prefixes and suffixes which, in combination with the INNs of Annex 3 to Regulation (EC) No 1549/2006, describe the salts, esters or hydrates of INNs; these salts, esters and hydrates are free of duty, on condition that they are classifiable in the same six-digit HS-subheading as the corresponding INN

Prefixes and suffixes can be combined (e.g. hydrochloride phosphate). They can be preceded by a multiplying prefix such as bi, bis, di, hemi, hepta, hexa, mono, penta, sesqui, tetra, tri, tris… (e.g. diacetate). Synonyms and systematic names can also be used, in the same way. INN means International Nonproprietary Names for pharmaceutical substances, World Health Organisation. INNRG means International Nonproprietary Names (INN) for pharmaceutical substances, Names for radicals & groups, comprehensive list 2004. INNCN means chemical or systematic name listed in International Nonproprietary Names (INN) for pharmaceutical substances, Names for radicals & groups, comprehensive list 2004. ID Preferred prefix or suffix Synonyms Systematic name when different 1 acefurate (INNRG) acetate (ester), furan-2-carboxylate (ester) (INNCN) 2 aceglumate (INNRG) rac-hydrogen N-acetylglutamate (INNCN) 3 aceponate (INNRG) acetate (ester), propanoate (ester) (INNCN) 4 acetate 5 acetonide (INNRG) propane-2,2-diylbis(oxy) (INNCN) 6 acetofenide acetophenide 1-phenylethane-1,1-diylbis(oxy) 7 1-acetoxyethyl 1-(acetyloxy)ethyl 8 aceturate (INNRG) N-acetylglycinate (INNCN) 10 acetylsalicylate 2-(acetyloxy)benzoate 11 acibutate (INNRG) acetate (ester), 2-methylpropanoate (ester) (INNCN) 12 acistrate (INNRG) acetate (ester), octadecanoate (ester) (INNCN) 13 acoxil (INNRG) (acetyloxy)methyl (INNCN) 14 adipate hexanedioate 15 alfoscerate (INNRG) (2R)-2,3-dihydroxypropyl hydrogen phosphate (INNCN) 16 alideximer (INNRG) poly([oxy(2-hydroxyethane-1,1-diyl)]{oxy[1-(hydroxymethyl)ethane-1,2-diyl]}) partly O-etherified with carboxymethyl groups with some carboxy groups amide linked to the tetrapeptide residue (glycylglycyl-L-phenylalanylglycyl) (INNCN) 17 allyl prop-2-en-1-yl 18 allylbromide allylobromide N-allyl, bromide (salt) 19 allyliodide allyloiodide N-allyl, iodide (salt) 20 aluminium 21 4-aminosalicylate aminosalicylate 2-hydroxy-4-aminobenzoate 22 ammonium 24 amsonate (INNRG) 2,2'-ethene-1,2-diylbis (5-aminobenzene-1-sulfonate) (INNCN) 25 anisatil (INNRG) 2-(4-methoxyphenyl)-2-oxoethyl (INNCN) 26 antipyrate 27 arbamel (INNRG) 2-(dimethylamino)-2-oxoethyl (INNCN) 28 argine (INNRG) 30Bα-L-arginine-30Bβ-L-arginine (INNCN) 29 arginine (INN) 30 aritox (INNRG) ricin A chain-MAB immunotoxine (INNCN) 31 ascorbate 32 aspart (INNRG) 28B-L-aspartic acid- (INNCN) 33 aspartate 34 axetil (INNRG) rac-1-(acetyloxy)ethyl (INNCN) 35 barbiturate 2,4,6(1H,3H,5H)-pyrimidinetrione 36 benetonide (INNRG) N-benzoyl-2-methyl-β-alanine (ester), acetonide (INNCN) 37 benzathine N,N'-dibenzylethylenediammonium 40 benzoacetate 41 benzoate (INNRG) 42 benzyl 43 benzylbromide benzylobromide N-benzyl, bromide (salt) 44 benzyliodide benzyloiodide N-benzyl, iodide (salt) 45 besilate (INNRG) besylate benzenesulfonate (INNCN), benzenesulphonate 47 bezomil (INNRG) (benzoyloxy)methyl (INNCN) 53 bismuth 55 borate 56 bromide (INNRG) 57 buciclate (INNRG) trans-4-butylcyclohexanecarboxylate (INNCN) 58 bunapsilate (INNRG) 3,7-di-tert-butylnaphthalene-1,5-disulfonate (INNCN) 59 buteprate (INNRG) butyrate (ester), propionate (ester) (INNCN) 60 butyl 62 tert-butyl t-butyl, tertiary butyl 67 butyl ester 69 tert-butyl ester t-butyl ester, tertiary butyl ester 75 butylbromide butylobromide N-butyl, bromide (salt) 76 butyrate butylate butanoate 77 calcium 82 camphorate 1,2,2-trimethyl-1,3-cyclopentanedicarboxylate 85 camsilate (INNRG) camsylate, camphorsulfonate, camphorsulphonate, R-camphorsulfonate, R-camphorsulphonate, S-camphorsulfonate, S-camphorsulphonate, camphor-10-sulfonate, camphor-10-sulphonate (7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl)methanesulfonate (INNCN) 87 caproate (INNRG) hexanoate (INNCN) 88 carbamate 89 carbesilate (INNRG) 4-sulfobenzoate (INNCN) 90 carbonate 91 chloride (INNRG) 95 choline (2-hydroxyethyl)trimethylammonium 96 ciclotate (INNRG) cyclotate 4-methylbicyclo[2.2.2]oct-2-ene-1-carboxylate (INNCN) 97 cilexetil (INNRG) rac-1-{[(cyclohexyloxy)carbonyl]oxy}ethyl (INNCN) 98 cinnamate 3-phenylprop-2-enoate 99 cipionate (INNRG) cypionate, cyclopentanepropionate 3-cyclopentylpropanoate (INNCN), 3-cyclopentylpropionate 100 citrate 2-hydroxypropane-1,2,3-tricarboxylate 101 cituxetan (INNRG) N-(4-{2(RS)-2-[bis(carboxymethyl)amino)]-3-({2-[bis(carboxymethyl)=amino]ethyl}(carboxymethyl)amino)propyl}phenyl)thiocarbamoyl (INNCN) 102 clofibrol (INNRG) 2-(4-chlorophenoxy)-2-methylpropyl (INNCN) 103 closilate (INNRG) closylate, p-chlorobenzenesulfonate, p-chlorobenzenesulphonate 4-chlorobenzene-1-sulfonate (INNCN), 4-chlorobenzenesulfonate 105 crobefate (INNRG) rac-{3-[(3E)-4-methoxybenzylidene]-2-(4-methoxyphenyl)chroman- 6-yl phosphate(2-)} (INNCN) 106 cromacate (INNRG) 2-[(6-hydroxy-4-methyl-2-oxo-2H-chromen-7yl)oxy]acetate (INNCN) 107 cromesilate (INNRG) (6,7-dihydroxy-2-oxo-2H-chromen-4-yl)methanesulfonate (INNCN) 108 crosfumaril (INNRG) (2E)-but-2-enedioyl (INNCN) 109 cyclamate (INNRG) N-cyclohexylsulfamate, N-cyclohexylsulphamate cyclohexylsulfamate (INNCN) 110a cyclohexylamine 111 cyclohexylammonium 112 cyclohexylpropionate cyclohexanepropionate cyclohexylpropanoate 118 daloxate (INNRG) L-alaninate (ester), (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (INNCN) 120 daropate (INNRG) dapropate 3-(dimethylamino)propanoate (INNCN) 121 deanil (INNRG) 2-(dimethylamino)ethyl (INNCN) 122 decanoate 123 decil (INNRG) decyl (INNCN) 124 defalan (INNRG) des-1B-L-phenylalanine-insulin (INNCN) 125 detemir (INNRG) tetradecanoyl (INNCN) 129 dibudinate (INNRG) 2,6-di-tert-butylnaphthalene-1,5-disulfonate (INNCN) 130 dibunate (INNRG) 2,6-di-tert-butylnaphthalene-1-sulfonate (INNCN) 133 dicibate (INNRG) dicyclohexylmethyl carbonate (INNCN) 134 dicyclohexylamine 135 dicyclohexylammonium 137 diethylamine 138 diethylammonium 139 diftitox (INNRG) N-L-methionyl-387-L-histidine-388-L-alanine-1-388-toxin (Corynebacterium diphtheriae strain C7) (388→2')-protein (INNCN) 142 digolil (INNRG) 2-(2-hydroxyethoxy)ethyl (INNCN) 149 dihydroxybenzoate 154 N,N-dimethyl-β-alanine N,N-dimethyl-beta-alanine 156 dinitrobenzoate 157 diolamine (INNRG) diethanolamine 2,2'-azanediyldiethanol (INNCN) 165 disulfide disulphide 169 docosil (INNRG) docosyl (INNCN) 170 dofosfate (INNRG) octadecyl hydrogen phosphate (INNCN) 171 ecamate (INNRG) N-ethylcarbamate (INNCN) 172 edamine (INNRG) ethane-1,2-diamine (INNCN) 173 edisilate (INNRG) edisylate, 1,2-ethanedisulfonate, 1,2-ethanedisulphonate ethane-1,2-disulfonate (INNCN) 175 embonate (INNRG) pamoate, 4,4'-methylenebis(3-hydroxy-2-naphthoate) 4,4'-methylenebis(3-hydroxynaphthalene-2-carboxylate) (INNCN) 176 enantate (INNRG) enanthate heptanoate (INNCN) 178 enbutate (INNRG) acetate (ester), butanoate (ester) (INNCN) 179 epolamine (INNRG) 1-pyrrolidineethanol 2-(pyrrolidin-1-yl)ethanol (INNCN) 180 erbumine (INNRG) tert-butylamine, t-butylamine, tertiary butylamine 2-methylpropan-2-amine (INNCN) 181 esilate (INNRG) esylate, ethanesulfonate, ethanesulphonate ethanesulfonate (INNCN) 182 estolate (INNRG) propionate dodecyl sulfate, propionate dodecyl sulphate, propionate lauryl sulfate, propionate lauryl sulphate propanoate (ester), dodecyl sulfate (salt) (INNCN) 184 etabonate (INNRG) ethyl carbonate (INNCN) 190 ethylbromide ethobromide N-ethyl, bromide (salt) 191 ethyl 192 ethyl ester 193 ethylamine 194 ethylammonium 195 ethylenantate ethylheptanoate 196 ethylenediamine ethane-1,2-diamine 197 ethylhexanoate 198 ethyliodide ethyloiodide N-ethyl, iodide (salt) 199 ethylsuccinate 200 etilsulfate (INNRG) ethylsulfate ethyl sulfate (INNCN) 201 farnesil (INNRG) (2E,6E)-3,7,11-trimethyldodeca-2,6,10-trien-1-yl (INNCN) 202 fendizoate (INNRG) 2-(6-hydroxybiphenyl-3-carbonyl)benzoate (INNCN) 203a ferrous 204 fluoride 205 fluorosulfonate fluorosulphonate 207 formate 209 fosfatex 210 fostedate (INNRG) tetradecyl hydrogen phosphate (INNCN) 211 fumarate (2E)-but-2-enedioate 212 furetonide (INNRG) 1-benzofurane-2-carboxylate (ester), propane-2,2-diylbis(oxy) (INNCN) 213 furoate furan-2(or 3)-carboxylate 213a fusidate 214 gadolinium 215 gamolenate (INNRG) (6Z,9Z,12Z)-octadeca-6,9,12-trienoate (INNCN) 216 glargine (INNRG) 21A-glycine-30Bα-L-arginine-30Bβ-L-arginine (INNCN) 217 glucarate saccharate (2R,3S,4S,5S)-2,3,4,5-tetrahydroxyhexanedioate, D-glucarate 218 gluceptate (INNRG) glucoheptonate D-glycero-D-gulo-heptonate (INNCN) 220 gluconate 221 glucoside 222 glulisine (INNRG) 3B-L-lysine,29B-L-glutamic acid (INNCN) 223 glutamer (INNRG) glutaraldehyde polymer (INNCN) 224 glycolate hydroxyacetate 225 glyoxylate oxoacetate 226 gold 227 guacil (INNRG) 2-methoxyphenyl (INNCN) 228 guanidine 230 hemisuccinate (INNRG) hydrogen succinate hydrogen butanedioate (INNCN) 235 hexacetonide (INNRG) 3,3-dimethylbutanoate (ester), propan-2,2-diylbis(oxy) (INNCN) 238 hibenzate (INNRG) hybenzate 4-(4-hydroxybenzoyl)benzoate (INNCN) 239 hippurate N-Benzoylglycine salt 241 hyclate (INNRG) ethanol — hydrogen chloride — water (0,5/1/0,5) (INNCN) 242 hydrate 243 hydrobromide 244 hydrochloride 248a hydrogen 261 hydroxide 262 hydroxybenzoate 263 2-(4-hydroxybenzoyl)benzoate o-(4-hydroxybenzoyl)benzoate 267 hydroxynaphtoate (INNRG) hydroxynaphthoate 3-hydroxynaphthalene-2-carboxylate (INNCN) 268 iodide (INNRG) 269 iodine-131 270 iron chloride 272 isetionate (INNRG) isethionate, 2-hydroxyethansulfonate, 2-hydroxyethansulphonate 2-hydroxyethane-1-sulfonate (INNCN) 273 isobutyrate 2-methylpropanoate 274 isocaproate 4-methylpentanoate 275 isonicotinate pyridine-4-carboxylate 276 isophthalate benzene-1,3-dicarboxylate 277 isopropionate 278 isopropyl propan-2-yl 279 lactate 2-hydroxypropanoate 280 lactobionate 4-O-(β-D-galactopyranosyl)-D-gluconate 281 laurate (INNRG) dodecanoate (INNCN) 282 lauril (INNRG) lauryl dodecyl (INNCN) 283 laurilsulfate (INNRG) lauril sulfate, lauril sulphate, lauryl sulfate, lauryl sulphate, laurilsulphate, laurylsulfate, laurylsulphate dodecyl sulfate (INNCN) 288 levulinate 4-oxopentanoate 289 lisetil (INNRG) L-lysinate (ester), diethyl (ester) (INNCN) 290 lisicol (INNRG) {N-[(5S)-5-carboxy-5-(3α,7α,12α-trihydroxy-5β-cholan-24-amido)pentyl]carbamothioyl}amino (INNCN) 291 lispro (INNRG) 28B-L-lysine-29B-L-proline (INNCN) 292 lithium 293 lutetium 294 lysinate lysine (INN) 296 mafenatox (INNRG) enterotoxin A (227-alanine) (Staphylococcus aureus) (INNCN) 297 magnesium 298 malate hydroxybutanedioate 299 maleate (Z)-but-2-enoate 300 malonate propanedioate 301 mandelate 2-hydroxy-2-phenylacetate, α-hydroxybenzeneacetate 302 medoxomil (INNRG) (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (INNCN) 303 megallate (INNRG) 3,4,5-trimethoxybenzoate (INNCN) 304 meglumine (INN) N-methylglucamine 1-deoxy-1-methylamino-D-glucitol 305 merpentan (INNRG) {N,N'-[1-(3-oxopropyl)ethane-1,2-diyl]bis(2-sulfanylacetamidato)}(4-) (INNCN) 306 mertansine (INNRG) tetrakis{(4RS)-4[(3-{[(1S)-2-{[(1S,2R,3S,5S,6S,16E,18E,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl]oxy}-1-methyl-2-oxoethyl]methylamino}-3-oxopropyl)disulfanyl]pentanoyl} (INNCN) 307 mesilate (INNRG) mesylate, methanesulfonate, methanesulphonate methanesulfonate (INNCN) 309 metembonate (INNRG) 4,4'-methylenebis(3-methoxynaphthalene-2-carboxylate) (INNCN) 312 methonitrate (INNRG) N-methyl, nitrate (salt) (INNCN) 313 methyl ester 315 methylbromide (INNRG) methobromide N-methyl, bromide (salt) (INNCN) 317 methylenedisalicylate methylenebis(2-hydroxybenzoate) 322 metilsulfate (INNRG) metilsulphate, methylsulfate, methylsulphate methyl sulfate (INNCN) 324 metiodide (INNRG) methyliodide N-methyl, iodide (salt) (INNCN) 325 mofetil (INNRG) 2-(morpholin-4-yl)ethyl (INNCN) 330 mucate galactarate, meso-galactarate 2,3,4,5-tetrahydroxyhexane-1,6-dioate 331 nafate formate sodium formyloxy (ester), sodium (salt) 332 napadisilate (INNRG) napadisylate, 1,5-naphthalenedisulfonate, 1,5-naphthalenedisulphonate naphthalene-1,5-disulfonate (INNCN) 338 napsilate (INNRG) napsylate, 2-naphthalenesulfonate, 2-naphthalenesulphonate naphthalene-2-sulfonate (INNCN) 340 nicotinate (INNRG) pyridine-3-carboxylate (INNCN) 341 nitrate 342 nitrobenzoate 343 octil (INNRG) octyl (INNCN) 344 olamine (INNRG) ethanolamine 2-aminoethanol (INNCN) 345 oleate (INNRG) (9Z)-octadec-9-enoate (INNCN) 346 orotate 1,2,3,6-tetrahydro-2,6-dioxopyrimidine-4-carboxylate 348 oxalate 349 oxide 351 oxoglurate (INNRG) hydrogen 2-oxopentanedioate (INNCN) 353 palmitate (INNRG) hexadecanoate (INNCN) 356 pantothenate N-(2,4-dihydroxy-3,3-dimethyl-1-oxobutyl)-β-alaninate 359 pegol (INNRG) α-(2-carboxyethyl)-ω-methoxypoly(oxyethane-1,2-diyl) (INNCN) 360 pendetide (INN) 362 pentexil (INNRG) pivetil (RS)-1-[(2,2-dimethylpropanoyl)oxy]ethyl (INNCN) 363 perchlorate (INNRG) 364 phenylpropionate 365 phosphate orthophosphate 366 phosphite 367 phthalate benzene-1,2-dicarboxylate 368 picrate 2,4,6-trinitrobenzene-1-olate 369 pivalate (INNRG) trimethylacetate 2,2-dimethylpropanoate (ester) (INNCN) 371 pivoxetil (INNRG) rac-1-[(2-methoxy-2-methylpropanoyl)oxy]ethyl (INNCN) 372 pivoxil (INNRG) (pivaloyloxy)methyl [(2,2-dimethylpropanoyl)oxy]methyl (INNCN) 374 poliglumex (INNRG) [poly(L-glutamic acid)z—(L-glutamate-γ-ester)—poly(L-glutamic acid)y]n (INNCN) 375 potassium (INNRG) potassium (INNCN) 378 propionate propanoate 383 propyl 384 propyl ester 385 proxetil (INNRG) rac-1-{[(propan-2-yloxy)carbonyl]oxy}ethyl (INNCN) 386 pyridylacetate pyridinylacetate 388 quinate 1,3,4,5-tetrahydroxycyclohexanecarboxylate 389 raffimer (INNRG) (2S,4R,6R,8S,11S,13S)-2,4,8,13-tetrakis(hydroxymethyl)-4,6,11-tris(ylomethyl)-3,5,7,10,12-pentaoxatetradecane-1,14-diyl (INNCN) 390 resinate abietate (1R,4aR,4bR,10aR)-1,4a-dimethyl-7-(1-methylethyl)-1,2,3,4,4a,4b,5,6,10,10a-decahydro-1-phenanthrenecarboxylate 392 salicylate (INNRG) 2-hydroxybenzoate (INNCN) 393 salicyloylacetate 2-hydroxybenzoylacetate 394 sesquioleate (INNRG) (9Z)-octadec-9-enoate(1,5) (INNCN) 395 sodium (INNRG) 413 soproxil (INNRG) {[(propan-2-yloxy)carbonyl]oxy}methyl (INNCN) 414 steaglate (INNRG) 2-(octadecanoyloxy)acetate (ester) (INNCN) 415 stearate (INNRG) octadecanoate (INNCN) 416 stinoprate (INNRG) N-acetylcysteinate (salt), propanoate (ester) (INNCN) 417 succinate butanedioate 418 succinil (INNRG) 3-carboxypropanoyl (INNCN) 419 succinyl butanedioyl 420 sudotox (INNRG) 248-L-histidine-249-L-methionine-250-L-alanine-251-L-glutamic acid-248-613-exotoxin A (Pseudomonas aeruginosa reduced) (INNCN) 421 suleptanate (INNRG) 8-[methyl(2-sulfoethyl)amino]-8-oxooctanoate (ester), monosodium salt (INNCN) 422 sulfate (INNRG) sulphate 423 sulfinate sulphinate 424 sulfite sulphite 424a sulfobenzoate sulphobenzoate 424b 3-sulfobenzoate 3-sulphobenzoate 425 sulfosalicylate sulphosalicylate 2-hydroxysulfobenzoate 426 sulfoxylate (INNRG) sulfinomethyl, monosodium salt (INNCN) 431 tafenatox (INNRG) enterotoxin A (Staphyloccus aureus) (INNCN) 432 tannate 433 tartrate (INNRG) L-tartrate (2R,3R)-2,3-dihydroxybutanedioate (INNCN), L-tartarate 434 D-tartrate (2S,3S)-2,3-dihydroxybutanedioate, D-tartarate 435 tebutate (INNRG) tert-butylacetate, t-butyl acetate, tertiary butyl acetate 3,3-dimethylbutanoate (INNCN) 436 tenoate (INNRG) thiophene-2-carboxylate (INNCN) 437 teoclate (INNRG) theoclate, 8-chlorotheophyllinate 8-chloro-1,3-dimethyl-2,6-dioxo-3,6-dihydro-1H-purin-7-(2H)-ide (INNCN) 438 teprosilate (INNRG) 3-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)propane-1-sulfonate (INNCN) 441 tetrahydrophthalate cyclohexene-1,2-dicarboxylate 444 tetraxetan (INNRG) [4,7,10-tris(carboxymethyl)-1,4,7,10-tetraazacyclodec-1-yl]acetyl (INNCN) 446 thiocyanate 447 tidoxil (INNRG) rac-2-(decyloxy)-3-(dodecylsulfanyl)propyl (INNCN) 448 tiuxetan (INNRG) N-(4-{(2S)-2-[bis(carboxymethyl)amino]-3-[(2RS)-{2-[bis(carboxymethyl)amino]propyl (carboxymethyl)amino]propyl} phenyl) thiocarbamoyl (INNCN) 449 tocoferil (INNRG) rac-(2R)-2,5,7,8-tetramethyl-2-[(4R,8R)-4,8,12-trimethyltridecyl]chroman-6-yl (INNCN) 450 tofesilate (INNRG) 3-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)ethane-1-sulfonate (INNCN) 453 tosilate (INNRG) tosylate, p-toluenesulfonate, p-toluenesulphonate 4-methylbenzene-1-sulfonate (INNCN) 455 triclofenate (INNRG) 2,4,5-trichlorophenolate (INNCN) 458 triflutate (INNRG) trifluoroacetate (INNCN) 463 trioleate (INNRG) tris[(9Z)-octadec-9-enoate] (INNCN) 465 tristearate (INNRG) tris(octadecanoate) (INNCN) 466 trolamine (INNRG) triethanolamine 2,2',2''-nitrilotriethanol (INNCN) 467 trometamol (INN) tromethamine 2-amino-2-(hydroxymethyl)propane-1,3-diol, tris(hydroxymethyl)methylamine 469 troxundate (INNRG) [2-(2-ethoxyethoxy)ethoxy]acetate (INNCN) 472 undecylate (INNRG) undecanoate (INNCN) 473 undecylenate (INNRG) undec-10-enoate (INNCN) 474 valerate (INNRG) pentanoate (INNCN) 475 xinafoate (INNRG) 1-hydroxynaphthalene-2-carboxylate (INNCN) 476 zinc

ANNEX III List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be added to the list of products receiving duty-free treatment included in Annex 6 to Regulation (EC) No 1549/2006

ID No CN code CAS RN Name 793 29021980 6746-94-7 ethynylcyclopropane 397 29052990 173200-56-1 (E)-6,6-dimethylhept-2-en-4-yn-1-ol 250 29055999 60827-45-4 (2S)-3-chloropropane-1,2-diol 320 29062900 127852-28-2 (1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethan-1-ol 308 29062900 167155-76-2 1,1-difluoro-1,1a,6,10b-tetrahydrodibenzo[a, e]cyclopropa[c][7]annulen-6-ol 530A 29093038 3259-03-8 1-(2-bromoethoxy)-2-ethoxybenzene or 2-bromoethyl 2-ethoxyphenyl ether 3 29093090 165254-21-7 1,2-bis{2-[2-(2-methoxyethoxy)ethoxy]ethoxy}-4,5-dinitrobenzene 124 29094990 170277-77-7 (3S)-3-[2-(mesyloxy)ethoxy]-4-(trityloxy)butyl methanesulfonate 636 29130000 80565-30-6 4'-chlorobiphenyl-4-carbaldehyde 566 29145000 17720-60-4 1-(2,4-dihydroxyphenyl)-2-(4-hydroxyphenyl)ethan-1-one 17 29145000 4495-66-3 1-[4-(benzyloxy)phenyl]propan-1-one 316 29145000 82499-20-5 (1R)-1-hydroxy-1-(3-hydroxyphenyl)acetone 712 29147000 124379-29-9 (4S)-4-(3,4-dichlorophenyl)-3,4-dihydronaphthalen-1(2H)-one 43 29147000 135306-45-5 1-(3,5-difluorophenyl)propan-1-one 59 29147000 162548-73-4 4,6-difluoroindan-1-one 158 29147000 190965-45-8 (2-bromo-5-propoxyphenyl)(2-hydroxy-4-methoxyphenyl)methanone 863 29147000 2196-99-8 2-chloro-1-(4-methoxyphenyl)ethan-1-one 314 29147000 2350-46-1 1-(2,3-dichloro-4-hydroxyphenyl)butan-1-one 827 29147000 26771-69-7 2-methoxy-1-[4-(trifluoromethyl)phenyl]ethan-1-one 550 29147000 43229-01-2 1-[4-(benzyloxy)-3-nitrophenyl]-2-bromoethan-1-one 64 29147000 62932-94-9 2-bromo-1-[4-hydroxy-3-(hydroxymethyl)phenyl]ethan-1-one 755 29153980 2243-35-8 2-oxo-2-phenylethyl acetate 519 29153980 60176-77-4 (1S,4R)-4-hydroxycyclopent-2-en-1-yl acetate 418 29155000 158894-67-8 1-bromo-2-methylpropyl propionate 796 29159020 7693-41-6 4-methoxyphenyl chloroformate 686 29162000 122665-97-8 4,4-difluorocyclohexane-1-carboxylic acid 937 29163900 114772-40-6 tert-butyl 4'-(bromomethyl)biphenyl-2-carboxylate 869 29163900 1716-12-7 sodium 4-phenylbutanoate 444 29163900 2444-36-2 (2-chlorophenyl)acetic acid 394 29163900 2901-13-5 ethyl 2-methyl-2-phenylpropanoate 67 29181985 111969-64-3 (1R,2S,5R)-2-isopropyl-5-methylcyclohexyl dihydroxyacetate or thymol glyoxylate 760 29181985 138-59-0 (3R,4S,5R)-3,4,5-trihydroxycyclohex-1-ene-1-carboxylic acid 544 29181985 20585-34-6 (2S)-cyclohexyl(hydroxy)phenylacetic acid 545 29181985 4335-77-7 cyclohexyl(hydroxy)phenylacetic acid 445 29181985 52950-18-2 (2R)-(2-chlorophenyl)hydroxyacetic acid 508 29183000 134176-18-4 ethyl 2-oxobicyclo[3.1.0]hexane-6-carboxylate 214 29183000 149437-76-3 5-(4-fluorophenyl)-5-oxopentanoic acid 21 29183000 39562-16-8 ethyl (E)-2-(3-nitrobenzylidene)-3-oxobutanoate 20 29183000 39562-22-6 2-methoxyethyl (E)-2-(3-nitrobenzylidene)-3-oxobutanoate 23 29183000 39562-27-1 methyl (2E)-2-(2-nitrobenzylidene)-3-oxobutanoate 315 29189990 1217-67-0 (4-butyryl-2,3-dichlorophenoxy)acetic acid 108 29189990 13335-71-2 (2,6-dimethylphenoxy)acetic acid 532 29189990 150726-89-9 dimethyl (2-methoxyphenoxy)malonate 402 29189990 204254-96-6 ethyl (1S,5R,6S)-5-(1-ethylpropoxy)-7-oxabicyclo[4.1.0]hept-3-ene-3-carboxylate 726 29209010 80841-78-7 4-(chloromethyl)-5-methyl-1,3-dioxol-2-one 436 29209085 163133-43-5 4-(nitrooxy)butyl (2S)-2-(6-methoxy-2-naphthyl)propanoate 540 29214980 259729-93-6 (1R)-1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutan-1-amine D-tartarate (1:1) 756 29214980 3789-59-1 (1S)-1-phenylpropan-1-amine 559 29214980 389056-74-0 (1S)-1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutan-1-amine D-tartarate (1:1) 558 29214980 84467-54-9 1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutan-1-amine 480 29215990 140-28-3 N, N'-dibenzylethane-1,2-diamine diacetate 226 29221980 114247-09-5 (3R)-N-methyl-3-phenyl-3-[4-(trifluoromethyl)phenoxy]propan-1-amine hydrochloride 84 29221980 115287-37-1 N-methyl-N-(4-nitrophenethyl)-2-(4-nitrophenoxy) ethan-1-amine 389 29221980 168960-19-8 ((1S,4R)-4-aminocyclopent-2-en-1-yl)methanol hydrochloride 669 29221980 214353-17-0 1-(2-amino-5-chlorophenyl)-2,2,2-trifluoroethane-1,1-diol hydrochloride 42 29221980 35320-23-1 (2R)-2-aminopropan-1-ol 512 29221980 42142-52-9 3-(methylamino)-1-phenylpropan-1-ol 670 29221980 467426-34-2 (2S)-2-(2-amino-5-chlorophenyl)-4-cyclopropyl-1,1,1-trifluorobut-3-yn-2-ol methanesulfonate (1:1.5) 547 29221980 56796-66-8 4-(benzyloxy)-α1-[(tert-butylamino)methyl]benzene-1,3-dimethanol 575 29221980 58997-87-8 2-(dimethylamino)-2-phenylbutan-1-ol 85 29222900 115256-13-8 4-(1-{[2-(4-aminophenoxy)ethyl]methylamino}ethyl)aniline 552 29222900 188690-84-8 (2S)-hydroxy(phenyl)acetic acid — (2R)-N-benzyl-1-(4-methoxyphenyl)propan-2-amine (1:1) (salt) 745 29222900 202197-26-0 3-chloro-4-[(3-fluorobenzyl)oxy]aniline 471 29223900 14189-82-3 (2E)-3-(N-methylanilino)acrylaldehyde 231 29224995 209216-09-1 2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid hydrate 857 29224995 223445-75-8 [(3S,4S)-1-(aminomethyl)-3,4-dimethylcyclopentyl]acetic acid 486 29224995 26774-89-0 sodium 2-(cyclohexa-1,4-dien-1-yl)-2-[((E)-1-methoxy-1-oxobut-2-en-2-yl)amino]acetate 549 29225000 174607-68-2 (1R)-1-[4-(benzyloxy)-3-(hydroxymethyl)phenyl]-2-(tert-butylamino)ethan-1-ol 48 29225000 196810-09-0 methyl N-(2-benzoylphenyl)-L-tyrosinate 548 29225000 50293-90-8 4-[(1R)-2-(tert-butylamino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol hydrochloride 860 29225000 62023-62-5 (2S,3S)-3-amino-2-hydroxy-4-phenylbutanoic acid 644 29225000 653574-13-1 methyl N-(benzyloxycarbonyl)valyl-D-alloisoleucylthreonylnorvalinate 945 29225000 71786-67-9 2-[benzyl(methyl)amino]-1-(3-hydroxyphenyl)ethan-1-one hydrochloride 18 29225000 96072-82-1 1-[4-(benzyloxy)phenyl]-2-[(4-phenylbutan-2-yl)amino]propan-1-one 379 29232000 4235-95-4 1,2-dioleoyl-sn-glycero-3-phosphocholine 377 29232000 77286-66-9 2-O-methyl-1-O-octadecyl-sn-glycero-3-phosphocholine 198 29241900 162537-11-3 N-(methoxycarbonyl)-3-methyl-L-valine 309 29241900 186193-10-2 (2S)-2-{[3-(tert-butoxycarbonyl)-2,2-dimethylpropanoyl]oxy}-4-methylpentanoic acid 378 29241900 228706-30-7 1,2-dioleoyl-sn-glycero-3-phospho[N-(4-carboxybutanoyl)ethanolamine] 12 29241900 89182-60-5 1-deoxy-1-formamidohexitol 352 29242995 132327-80-1 N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-N5-trityl-L-glutamine 348 29242995 132388-59-1 N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-N4-trityl-L-asparagine 183 29242995 170361-49-6 N-(3,4-dichlorophenyl)-N-{3-[(2,3-dihydroinden-2-yl)methylamino]propyl}-5,6,7,8-tetrahydronaphthalene-2-carboxamide 102 29242995 194085-75-1 2-(2-chlorophenyl)-2-hydroxyethyl carbamate 398 29242995 22871-58-5 3-amino-5-[(2-hydroxyethyl)carbamoyl]-2,4,6-triiodobenzoic acid 360 29242995 244191-94-4 N-[(9H-fluoren-9-ylmethoxy)carbonyl]-α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucine, 1,4,6,9-tetra-tert-butyl ester 13 29242995 28197-66-2 N-[3-acetyl-4-(oxiran-2-ylmethoxy)phenyl]butanamide 687 29242995 325715-13-7 N-(3-acetylphenyl)-N-methylacetamide 347 29242995 35661-39-3 N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanine 349 29242995 35661-60-0 N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-leucine 598 29242995 376348-76-4 ethyl (3S)-3-(4,4-difluorocyclohexane-1-carboxamido)-3-phenylpropanoate 599 29242995 376348-77-5 4,4-difluoro-N-((1S)-3-hydroxy-1-phenylpropyl)cyclohexane-1-carboxamide 600 29242995 376348-78-6 4,4-difluoro-N-((1S)-3-oxo-1-phenylpropyl)cyclohexane-1-carboxamide 619 29242995 40371-50-4 (2S)-4-{[(benzyloxy)carbonyl]amino}-2-hydroxybutanoic acid 731 29242995 481659-97-6 tert-butyl {(1S)-2-[benzyl(methyl)amino]-2-oxo-1-phenylethyl}carbamate hydrochloride 411 29242995 49705-98-8 benzyl ((1S,2R)-1-carbamoyl-2-hydroxypropyl)carbamate 144 29242995 53947-84-5 2-(carboxyacetamido)benzoic acid 487 29242995 6485-67-2 (2R)-2-amino-2-phenylacetamide 371 29242995 65864-22-4 L-phenylalaninamide 696 29242995 667937-05-5 3-[4-(trifluoromethyl)anilino]pentanamide 350 29242995 71989-14-5 4-tert-butyl N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-aspartate 351 29242995 71989-18-9 5-tert-butyl N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-glutamate 353 29242995 71989-20-3 N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-glutamine 355 29242995 71989-23-6 N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-isoleucine 356 29242995 71989-26-9 N6-(tert-butoxycarbonyl)-N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-lysine 367 29242995 71989-33-8 O-tert-butyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-serine 368 29242995 71989-35-0 O-tert-butyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-threonine 370 29242995 71989-38-3 O-tert-butyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-tyrosine 412 29242995 80082-51-5 3-amino-2-{[(benzyloxy)carbonyl]amino}-1-methyl-3-oxopropyl methanesulfonate 197 29242995 98760-08-8 tert-butyl [1-((2S)-oxiran-2-yl)-2-phenylethyl]carbamate 317 29252900 249561-98-6 tris{[(2Z)-2-chloro-3-(dimethylamino)prop-2-en-1-ylidene]dimethylammonium} hexafluorophosphate(3-) 215 29252900 3382-63-6 4-{(E)-[(4-fluorophenyl)imino]methyl}phenol 938 29269095 114772-54-2 4'-(bromomethyl)biphenyl-2-carbonitrile 142 29269095 152630-47-2 1-[3-(cyclopentyloxy)-4-methoxyphenyl]-4-oxocyclohexane-1-carbonitrile 143 29269095 152630-48-3 dimethyl 4-cyano-4-[3-(cyclopentyloxy)-4-methoxyphenyl]heptanedioate 585 29269095 192869-10-6 2-iodo-3,4-dimethoxy-6-nitrobenzonitrile 586 29269095 192869-24-2 6-amino-2-iodo-3,4-dimethoxybenzonitrile 539 29269095 28049-61-8 1-(4-chlorophenyl)cyclobutane-1-carbonitrile 528 29269095 31915-40-9 N-[1-cyano-2-(4-hydroxyphenyl)-1-methylethyl]acetamide 673 29269095 474645-97-1 (3R)-3-aminopentanenitrile methanesulfonate 803 29269095 604784-44-3 tert-butylammonium (Z)-3-cyano-5-methylhex-3-enoate 287 29280090 212631-79-3 2-(2-chloro-4-iodoanilino)-N-(cyclopropylmethoxy)-3,4-difluorobenzamide 33 29280090 253605-31-1 N-hydroxy-2-methylpropan-2-amine acetate (salt) or tert-butylhydroxylamine acetate (salt) 49 29280090 618-26-8 1-methyl-1-phenylhydrazine sulfate (2:1) 403 29299000 204254-98-8 ethyl (3R,4S,5R)-5-azido-3-(1-ethylpropoxy)-4-hydroxycyclohex-1-ene-1-carboxylate 405 29299000 204255-06-1 ethyl (3R,4R,5S)-4-acetamido-5-azido-3-(1-ethylpropoxy)cyclohex-1-ene-1-carboxylate 748 29309085 104458-24-4 2-mesylethan-1-amine hydrochloride 399 29309085 153277-33-9 methyl N-[(benzyloxy)carbonyl]-S-phenyl-L-cysteinate 862 29309085 15570-12-4 3-methoxybenzene-1-thiol 56 29309085 16188-55-9 [4-(methylsulfanyl)phenyl]acetic acid 26 29309085 225652-11-9 1-(4-chlorophenoxy)-4-(methylsulfanyl)benzene or 4-chlorophenyl 4-(methylsulfanyl)phenyl ether 339 29309085 2736-23-4 2,4-dichloro-5-mesylbenzoic acid 595 29309085 289717-37-9 N, N-dimethyl-2-[4-(methylsulfanyl)phenoxy]benzylamine hydrochloride 742 29309085 346413-00-1 1-(4-ethoxyphenyl)-2-(4-mesylphenyl)ethan-1-one 358 29309085 3483-12-3 (2R,3S)-1,4-disulfanylbutane-2,3-diol or dithiothreitol 594 29309085 364323-64-8 2-[4-(methylsulfanyl)phenoxy]benzaldehyde 864 29309085 40248-84-8 3-sulfanylphenol 324 29309085 50413-24-6 2-bromo-1-(4-mesylphenyl)ethan-1-one 65 29309085 90536-66-6 (4-mesylphenyl)acetic acid 206 29310095 123599-82-6 {[2-methyl-1-(propionyloxy)propoxy](4-phenylbutyl)phosphoryl}acetic acid 58 29310095 27784-76-5 tert-butyl (diethoxyphosphoryl)acetate 789 29310095 649761-22-8 (1R,5S)-5-[dimethyl(phenyl)silyl]-2-(hydroxymethyl)cyclopent-2-ene-1-carboxylic acid — (1R,2R)-2-amino-1-(4-nitrophenyl)propane-1,3-diol (1:1) (salt) 391 29310095 86552-32-1 (4-phenylbutyl)phosphinic acid 747 29321900 27329-70-0 (5-formyl-2-furyl)boronic acid 762 29321900 37076-71-4 1,2,3-tri-O-acetyl-5-deoxy-D-ribofuranose 700 29321900 87392-07-2 (2S)-tetrahydrofuran-2-carboxylic acid 582 29322985 122111-01-7 [(2R)-2-(benzoyloxy)-4,4-difluoro-5-oxotetrahydrofuran-2-yl]methyl benzoate 78 29322985 142680-85-1 (25S)-25-cyclohexyl-25-de(sec-butyl)-5-O-demethyl-22,23-dihydroavermectin A1a 244 29322985 145667-75-0 (3aR,4R,5R,6aS)-5-hydroxy-4-((3R)-3-hydroxy-5-phenylpentyl)hexahydrocyclopenta[b]furan-2-one 79 29322985 220119-16-4 (25S)-cyclohexyl-25-de(sec-butyl)- 5-demethoxy-5-oxo-22,23-dihydroavermectin A1a 942 29322985 221129-55-1 (6R)-4-hydroxy-6-phenethyl-6-propyl-5,6-dihydro-2H-pyran-2-one 115 29322985 51559-36-5 5-methoxy-2H-chromen-2-one 660 29322985 95716-70-4 7α-(methoxycarbonyl)-3-oxo-17α-pregna-4,9(11)-diene-21,17-carbolactone 703 29322985 96829-59-3 (1S,3E,6E)-1-[((2S,3S)-3-hexyl-4-oxooxetan-2-yl)methyl]dodeca-3,6-dien-1-yl N-formyl-L-leucinate 37 29329970 124655-09-0 tert-butyl [(4R,6S)-6-(hydroxymethyl)-2,2-dimethyl-1,3-dioxan-4-yl]acetate 567 29329970 130064-21-0 1-{2-hydroxy-4-[(tetrahydropyran-2-yl)oxy]phenyl}-2-{4-[(tetrahydropyran-2-yl)oxy]phenyl}ethan-1-one 156 29329970 167256-05-5 methyl (1S,2S)-1-(1,3-benzodioxol-5-yl)-3-(2-hydroxy-4-methoxyphenyl)-5-propoxyindane-2-carboxylate 157 29329970 191106-49-7 methyl (1S,2S)-1-(1,3-benzodioxol-5-yl)-3-[2-(benzyloxy)-4-methoxyphenyl]-5-propoxyindane-2-carboxylate 189 29329970 192201-93-7 2-({3-[5-(6-methoxy-1-naphthyl)-1,3-dioxan-2-yl]propyl}methylamino)-N-methylacetamide 127 29329970 196303-01-2 (7S)-7-methyl-5-(4-nitrophenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isochromene 62 29329970 7772-94-3 2-acetamido-2-deoxy-β-D-mannopyranose 607 29329985 115437-18-8 (2α,4α,5β,7β,10β,13β)-4-acetoxy-1,10,13-trihydroxy-9-oxo-7-[(triethylsilyl)oxy]-5,20-epoxytax-11-en-2-yl benzoate 608 29329985 115437-21-3 (4α)-4,10-diacetoxy-1,13-dihydroxy-9-oxo-7-[(triethylsilyl)oxy]-5,20-epoxytax-11-en-2-yl benzoate 54 29329985 130525-58-5 methyl 5-acetamido-7,8,9-O-triacetyl-2,6-anhydro-4-azido-3,4,5-trideoxy-D-glycero-D-galacto-non-2-enonate 609 29329985 149107-93-7 (2α,4α,5β,7β,10β,13α)-4,10-diacetoxy-13-{[(2R,3S)-3-benzamido-2-(1-methoxy-1-methylethoxy)-3-phenylpropanoyl]oxy}-1-hydroxy-9-oxo-7-[(triethylsilyl)oxy]-5,20-epoxytax-11-en-2-yl benzoate 652 29329985 199796-52-6 (2α,4α,7β,10β,13α)-4,10-diacetoxy-13-({(2R,3S)-3-benzamido-2-[((4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoyl)oxy]-3-phenylpropanoyl}oxy)-1,7-dihydroxy-9-oxo-5,20-epoxytax-11-en-2-yl benzoate 11 29329985 65293-32-5 N-β-D-glucopyranosylformamide 590 29331990 334828-10-3 4-amino-5-ethyl-1-(2-methoxyethyl)pyrazole-3-carboxamide 511 29332100 186462-71-5 (1R,2R,5S,6R)-2',5'-dioxospiro[bicyclo[3.1.0]hexane-2,4'-imidazolidine]-6-carboxylic acid 354 29332990 109425-51-6 N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-N-trityl-L-histidine 263 29332990 178982-67-7 2-[(benzyloxy)methyl]-4-isopropylimidazole 359 29332990 244191-88-6 N-acetyl-O-tert-butyl-L-tyrosyl-O-tert-butyl-L-threonyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-N1-trityl-L-histidyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-α-L-glutamyl-α-L-glutamyl-O-tert-butyl-L-seryl-N-trityl-L-glutaminyl-N-trityl-L-asparaginyl-N-trityl-L-glutaminyl-L-glutamine, 10,11-di-tert-butyl ester 365 29332990 244244-26-6 N-acetyl-O-tert-butyl-L-tyrosyl-O-tert-butyl-L-threonyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-N1- trityl-L-histidyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-α-L-glutamyl-α-L-glutamyl-O-tert-butyl-L-seryl-N-trityl-L-glutaminyl-N-trityl-L-asparaginyl-N-trityl-L-glutaminyl-L-glutaminyl-α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucyl-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, hepta-tert-butyl ester 583 29332990 68283-19-2 (2-butylimidazol-5-yl)methanol 954 29333999 0-00-0 11-ethyl-5-methyl-8-{2-[(1-oxo-1λ4-quinolin-4-yl)oxy]ethyl}-11H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6(5H)-one 119 29333999 100238-42-4 4-(2-piperidin-1-ylethoxy)phenol 541 29333999 103129-82-4 3-ethyl 5-methyl 2-[(2-aminoethoxy)methyl]-4-(2-chlorophenyl)-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate 167 29333999 127293-57-6 (1R)-1-(4-chlorophenyl)-2-[4-(4-fluorobenzyl)piperidin-1-yl]ethan-1-ol 16 29333999 158878-47-8 (3R,5R)-3-{(E)-2-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]vinyl}-5-hydroxycyclohexan-1-one 14 29333999 159813-78-2 (3R,5S,6E)-7-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]-3,5-dihydroxyhept-6-enoic acid 621a 29333999 161417-03-4 2-methyl-3-((2S)-pyrrolidin-2-ylmethoxy)pyridine 9 29333999 177964-68-0 3-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]acrylaldehyde 168 29333999 178460-82-7 (1R)-1-(4-chlorophenyl)-2-[4-(4-fluorobenzyl)piperidin-1-yl]ethan-1-ol hydrochloride 264 29333999 178981-89-0 {5-[(3,5-dichlorophenyl)sulfanyl]-4-isopropyl-1-(pyridin-4-ylmethyl)imidazol-2-yl}methanol 173 29333999 188396-54-5 1-(2-biphenyl-4-ylethyl)-4-[3-(trifluoromethyl)phenyl]-1,2,3,6-tetrahydropyridine hydrochloride 875 29333999 19395-39-2 2-phenyl-2-piperidin-2-ylacetamide 196 29333999 198904-85-7 tert-butyl 2-(4-pyridin-2-ylbenzyl)hydrazine-1-carboxylate 199 29333999 198904-86-8 tert-butyl 2-{(2S,3S)-3-[(tert-butoxycarbonyl)amino]-2-hydroxy-4-phenylbutyl}-2-[4-(pyridin-2-yl)benzyl]hydrazine-1-carboxylate 840 29333999 213839-64-6 N-{2-[5-(aminoiminomethyl)-2-hydroxyphenoxy]-3,5-difluoro-6-[3-(1-methyl-4,5-dihydroimidazol-2-yl)phenoxy]pyridin-4-yl]-N-methyglycine dihydrochloride 442 29333999 221180-26-3 4-amino-5-chloro-2-methoxy-N-(3-methoxypiperidin-4-yl)benzamide 318 29333999 221615-75-4 2-(4-mesylphenyl)-1-(6-methylpyridin-3-yl)- ethan-1-one 690 29333999 230615-52-8 2,3,4,5-tetrahydro-1H-1,5-methano-3-benzazepine hydrochloride 661 29333999 230615-59-5 7,8-dinitro-3-(trifluoroacetyl)-2,3,4,5-tetrahydro-1H-1,5-methano-3-benzazepine 765 29333999 25333-42-0 (3R)-quinuclidin-3-ol 565 29333999 26815-04-3 4-(2-piperidin-1-ylethoxy)benzaldehyde 842 29333999 280129-82-0 4-({2-[(benzyloxy)methyl]-4-isopropylimidazol-1-yl}methyl)pyridine oxalate (1:2) 490 29333999 319460-85-0 N-methyl-2-{[3-((E)-2-pyridin-2-ylvinyl)-1H-indazol-6-yl]sulfanyl}benzamide 489 29333999 319460-94-1 N-(2-fluoro-5-{[3-((E)-2-pyridin-2-ylvinyl)-1H-indazol-6-yl]amino}phenyl)-1,3-dimethylpyrazole-5-carboxamide 579 29333999 37699-43-7 2,3-dimethyl-4-nitropyridine 1-oxide 210 29333999 4021-07-2 3-methylpyridine-2-carboxylic acid 649 29333999 423165-13-3 8-benzyl-3-exo-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)-8-azabicyclo[3.2.1]octane 951 29333999 429659-01-8 ethyl N-[4-(methylamino)-3-nitrobenzoyl]-N-pyridin-2-yl-ß-alaninate 560 29333999 43200-82-4 6-(5-chloropyridin-2-yl)-5H-pyrrolo[3,4-b]pyrazine-5,7(6H)-dione 564 29333999 440634-25-3 tert-butyl 4-{2-[4-(mesyloxy)piperidin-1-yl]-2-oxoethyl}piperidine-1-carboxylate 538 29333999 58859-46-4 ethyl 4-aminopiperidine-1-carboxylate 626 29333999 78750-68-2 4-[(3-aminopyridin-2-yl)amino]phenol 513 29333999 84449-81-0 4-(2-piperidin-1-ylethoxy)benzoyl chloride hydrochloride 948 29334990 0-00-0 2-(ethylamino)-5-[2-(quinolin-4-yloxy)ethyl]nicotinic acid 483 29334990 10500-57-9 5,6,7,8-tetrahydroquinoline 149 29334990 106635-86-3 2,6-dimethoxy-4-methyl-5-[3-(trifluoromethyl)phenoxy]quinolin-8-amine 647 29334990 118864-75-8 (1S)-1-phenyl-1,2,3,4-tetrahydroisoquinoline 36 29334990 172649-40-0 3-[(4S)-5-oxo-2-(trifluoromethyl)-1,4,5,6,7,8-hexahydroquinolin-4-yl]benzonitrile 623 29334990 189279-58-1 1-(6-amino-3,5-difluoropyridin-2-yl)-8-chloro-6-fluoro-7-(3-hydroxyazetidin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid 150 29334990 189746-15-4 2,6-dimethoxy-4-methyl-8-nitro-5-[3-(trifluoromethyl)phenoxy]quinoline 152 29334990 189746-19-8 5-chloro-2,6-dimethoxy-4-methylquinoline 151 29334990 189746-21-2 5-chloro-2,6-dimethoxy-4-methyl-8-nitroquinoline 434 29334990 194804-45-0 ethyl 1-cyclopropyl-8-(difluoromethoxy)-7-((1R)-1-methyl-2-tritylisoindolin-5-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate 433 29334990 194805-07-7 ethyl 7-bromo-1-cyclopropyl-8-(difluoromethoxy)-4-oxo-1,4-dihydroquinoline-3-carboxylate 705A 29334990 209909-03-5 (2-chloro-6,7-difluoroquinolin-3-yl)methanol 704A 29334990 220998-08-3 {2,7-dichloro-6-methyl-4-[(4-methylpiperidin-1-yl)methyl]quinolin-3-yl}methanol 386 29334990 287930-77-2 (1S)-1-{3-[(E)-2-(7-chloroquinolin-2-yl)vinyl]phenyl}-3-[2-(1-hydroxy-1-methylethyl)phenyl]propan-1-ol 387 29334990 287930-78-3 methyl 2-((3S)-3-{3-[(E)-2-(7-chloroquinolin-2-yl)vinyl]phenyl}-3-hydroxypropyl)benzoate hydrate 674 29334990 474645-93-7 methyl [2-ethyl-6-(trifluoromethyl)-1,2,3,4-tetrahydroquinolin-4-yl]carbamate 153 29334990 6340-55-2 2,6-dimethoxy-4-methylquinoline 664 29334990 79276-06-5 tert-butyl (3S)-1,2,3,4-tetrahydroisoquinoline-3-carboxylate 4-methylbenzenesulfonate 455 29335995 119532-26-2 1-(2,3-dichlorophenyl)piperazine 80 29335995 137234-74-3 4-chloro-6-ethyl-5-fluoropyrimidine 509 29335995 137281-39-1 4-[2-(2-amino-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoic acid 39 29335995 140373-09-7 4-{[(3-{[(2,2-dimethylpropanoyl)oxy]methyl}-2,7-dimethyl-4-oxo-3,4-dihydroquinazolin-6-yl)methyl](prop-2-yn-1-yl)amino}-2-fluorobenzoic acid 531 29335995 14080-23-0 pyrimidine-2-carbonitrile 38 29335995 160009-37-0 methyl 4-(4-fluorophenyl)-6-isopropyl-2-(N-methylmethanesulfonamido)]pyrimidine-5-carboxylate 744 29335995 16064-08-7 6-iodoquinazolin-4(1H)-one 123 29335995 167465-36-3 (2R)-1-[4-((1aR,10bS)-1,1-difluoro-1,1a,6,10b-tetrahydrodibenzo[a, e]cyclopropa[c][7]annulen-6-yl)piperazin-1-yl]-3-[(quinolin-5-yl)oxy]propan-2-ol trihydrochloride 73 29335995 188416-20-8 3-(6-chloro-5-fluoropyrimidin-4-yl)-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butan-2-ol hydrochloride 81 29335995 188416-28-6 4-(1-bromoethyl)-6-chloro-5-fluoropyrimidine 112 29335995 192725-50-1 (2S)-3-methyl-2-(2-oxohexahydropyrimidin-1-yl)butanoic acid 133 29335995 192726-06-0 (2S)-N-[(1S,3S,4S)-4-amino-1-benzyl-3-hydroxy-5-phenylpentyl]-3-methyl-2-(2-oxotetrahydropyrimidin-1(2H)-yl)butanamide — 5-oxopyrrolidine-2-carboxylic acid (1:1) (salt) 790 29335995 19916-73-5 6-(benzyloxy)-9H-purin-2-amine 261 29335995 214287-88-4 (4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluoromethyl)-3,4-dihydroquinazolin-2(1H)-one 259 29335995 214287-99-7 (4S)-6-chloro-4-((E)-2-cyclopropylvinyl)-4-(trifluoromethyl)-3,4-dihydroquinazolin-2(1H)-one 653 29335995 225916-82-5 8-chloro-5-((4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoyl)-11-(4-methylpiperazin-1-yl)-5H-dibenzo[b, e][1,4]diazepine 746 29335995 231278-20-9 N-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-iodoquinazolin-4-amine 256 29335995 247565-04-4 (4S)-6-chloro-4-(cyclopropylethynyl)-3-((R)-1-phenylethyl)-4-(trifluoromethyl)-3,4-dihydroquinazolin-2(1H)-one 554 29335995 345217-02-9 1-[(1S,2S)-2-(benzyloxy)-1-ethylpropyl]-N-{4-[4-(4-hydroxyphenyl)piperazin-1-yl]phenyl}hydrazine-1-carboxamide 313 29335995 487-21-8 pteridine-2,4(1H,3H)-dione 958 29335995 518048-03-8 2-(1-amino-1-methylethyl)-N-(4-fluorobenzyl)-5-hydroxy-1-methyl-6-oxo-1,6-dihydropyrimidine-4-carboxamide 949 29335995 57061-71-9 1-(2-chloroethyl)-4-[3-(trifluoromethyl)phenyl]piperazine dihydrochloride 561 29335995 59878-63-6 6-(5-chloropyridin-2-yl)-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazin-5-yl piperazine-1-carboxylate 830 29335995 599179-03-0 1-(4,6-dimethylpyrimidine-5-carbonyl)- 4-((3S)-4-{(1R)-2-methoxy-1-[4-(trifluoromethyl)phenyl]ethyl}-3-methylpiperazin-1-yl)-4-methylpiperidine maleate (1:1) 828 29335995 612494-10-7 1-{(1R)-2-methoxy-1-[4-(trifluoromethyl)phenyl]ethyl}-2-methylpiperazine D-tartarate (1:1) 829 29335995 612543-01-8 1-(4,6-dimethylpyrimidine-5-carbonyl)piperidin-4-one 791 29335995 649761-23-9 (1S,2S,3S,5S)-5-[2-amino-6-(benzyloxy)-9H-purin-9-yl]-2-[(benzyloxy)methyl]-3-[dimethyl(phenyl)silyl]-1-(hydroxymethyl)cyclopentan-1-ol 792 29335995 649761-24-0 2-amino-9-{(1S,3R,4S)-3-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]-2-methylidenecyclopentyl}-9H-purin-6(1H)-one 835 29335995 654671-77-9 (2R)-4-oxo-4-[3-(trifluoromethyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine phosphate (1:1) hydrate 946 29335995 7139-02-8 2,6-dichloro-4,8-dipiperidinopyrimido[5,4-d]pyrimidine 457 29337900 105318-28-3 ((2S,3S)-2-{(1R)-2-[(4-chlorophenyl)sulfanyl]-1-methyl-2-oxoethyl}-3-((1R)-1-hydroxyethyl)-4-oxoazetidin-1-yl)acetic acid 610 29337900 133066-59-8 (3R,4S)-2-oxo-4-phenylazetidin-3-yl acetate 60 29337900 148776-18-5 (2-oxo-1-phenylpyrrolidin-3-yl)triphenylphosphonium bromide 612 29337900 149107-92-6 1-benzoyl-3-(1-methoxy-1-methylethoxy)-4-phenylazetidin-2-one 692 29337900 162142-14-5 1-cyclopentyl-3-ethyl-1,4,5,6-tetrahydro-7H-pyrazolo[3,4-c]pyridin-7-one 50 29337900 198213-15-9 sodium 3-(methoxycarbonyl)-2-oxo-1,2,5,6-tetrahydropyridin-4-olate 188 29337900 205881-86-3 6-fluoro-9-methyl-2-phenyl-4-(pyrrolidine-1-carbonyl)-9H-pyrido[3,4-b]indol-1(2H)-one 176 29337900 244080-24-8 1-ethyl-9-methoxy-2,6,7,12-tetrahydroindolo[2,3-a]quinolizin-4(3H)-one 491 29337900 283173-50-2 8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one 693 29337900 303752-13-8 1-cyclopentyl-3-ethyl-6-(4-methoxybenzyl)-1,4,5,6-tetrahydro-7H-pyrazolo[3,4-c]pyridin-7-one 4-methylbenzene-1-sulfonate 148 29337900 3197-25-9 2-(4-oxopentyl)-1H-isoindole-1,3(2H)-dione 776 29337900 341031-54-7 N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethylpyrrole-3-carboxamide L-malate (1:1) 713 29337900 43200-81-3 6-(5-chloropyridin-2-yl)-7-hydroxy-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazin-5-one 154 29337900 5342-23-4 6-methoxy-4-methylquinolin-2(1H)-one 413 29337900 80082-62-8 tetrabutylammonium (2S,3S)-3-{[(benzyloxy)carbonyl]amino}-2-methyl-4-oxoazetidine-1-sulfonate 414 29337900 80082-65-1 (2S,3S)-3-amino-2-methyl-4-oxoazetidine-1-sulfonic acid 140 29339940 193077-87-1 [(2S)-7-(2-methoxy-2-oxoethyl)-4-methyl-3-oxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-yl]acetic acid 139 29339940 210288-67-8 [(2S)-7-iodo-4-methyl-3-oxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-yl]acetic acid 392 29339990 103201-78-1 4-cyclohexylproline 120 29339990 113963-68-1 3,4-di(indol-3-yl)-1-methylpyrrole-2,5-dione 322 29339990 119192-10-8 4-[(1H-1,2,4-triazol-1-yl)methyl]aniline 422 29339990 120807-02-5 (4S)-N-benzoyl-4-(mesyloxy)-L-proline 369 29339990 143824-78-6 N1-(tert-butoxycarbonyl)-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-tryptophan 227 29339990 14907-27-8 methyl D-tryptophanate hydrochloride 4 29339990 149365-59-3 dibenzyl 5,5'-[(3,4-diethylpyrrole-2,5-diyl)bis(methylene)]bis[4-(3-methoxy-3-oxopropyl)-3-methylpyrrole-2-carboxylate] 5 29339990 149365-62-8 5,5'-[(3,4-diethylpyrrole-2,5-diyl)bis(methylene)]bis[4-(3-hydroxypropyl)-3-methylpyrrole-2-carbaldehyde] 940 29339990 152628-02-9 1,4'-dimethyl-2'-propyl-1H,1'H-2,6'-bibenzimidazole 939 29339990 152628-03-0 4-Methyl-2-propylbenzimidazole-6-carboxylic acid 323 29339990 160194-39-8 2-{5-[(1H-1,2,4-triazol-1-yl)methyl]indol-3-yl}ethan-1-ol 312 29339990 16298-03-6 methyl 3-aminopyrazine-2-carboxylate 35 29339990 171964-73-1 [N-(4-methoxybenzoyl)-L-valyl]-N-[(1S)-3,3,3-trifluoro-1-isopropyl-2-oxopropyl]-L-prolinamide 230 29339990 172733-42-5 sodium [(1-benzyl-2-ethyl-3-oxamoylindol-4-yl)oxy]acetate 87 29339990 180637-89-2 3-[((2R)-1-methylpyrrolidin-2-yl)methyl]-5-[(E)-2-(phenylsulfonyl)vinyl]indole 677 29339990 180915-94-0 1-{2-[4-(6-methoxy-3,4-dihydro-1-naphthyl)phenoxy]ethyl}pyrrolidine 676 29339990 180915-95-1 1-{2-[4-(2-bromo-6-methoxy-3,4-dihydro-1-naphthyl)phenoxy]ethyl}pyrrolidine 31 29339990 181827-47-4 [N-(methoxycarbonyl)-L-valyl]-L-proline 86 29339990 188113-71-5 1-acetyl-3-[((2R)-1-methylpyrrolidin-2-yl)methyl]-5-[(E)-2-(phenylsulfonyl)vinyl]indole 27 29339990 193274-37-2 3a-benzyl-2-methyl-2,3a,4,5,6,7-hexahydro-3H-pyrazolo[4,3-c]pyridin-3-one L-tartarate 137 29339990 197143-35-4 (3Z)-4-(aminomethyl)pyrrolidin-3-one O-methyloxime dihydrochloride 404 29339990 204255-02-7 ethyl (1R,5R,6R)-5-(1-ethylpropoxy)-7-azabicyclo[4.1.0]hept-3-ene-3-carboxylate 794 29339990 210558-66-0 (1R,2S)-1-phenyl-2-pyrrolidin-1-ylpropan-1-ol hydrochloride 319 29339990 219909-83-8 3-((4S)-4-sulfanyl-L-prolinamidol)benzoic acid hydrochloride 634 29339990 221030-56-4 2-(4-fluorophenyl)-4-(3-hydroxy-3-methylbutoxy)-5-(4-mesylphenyl)pyridazin-3(2H)-one 743 29339990 221148-46-5 2-(4-ethoxyphenyl)-3-(4-mesylphenyl)pyrazolo[1,5-b]pyridazine 245 29339990 227025-33-4 1-benzyl-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one 441 29339990 235106-62-4 2,2'-[(4-hydroxyphenyl)methylene]bis(4-{(E)-[(5-methyl-1H-tetrazol-1-yl)imino]methyl}phenol) 362 29339990 244191-95-5 α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, tert-butyl ester 361 29339990 244191-96-6 N-[(9H-fluoren-9-ylmethoxy)carbonyl]-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophan, 1-tert-butyl ester 363 29339990 244244-29-9 N-[(9H-fluoren-9-ylmethoxy)carbonyl]-α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucyl-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, penta-tert-butyl ester 364 29339990 244244-31-3 α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucyl-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, penta-tert-butyl ester monohydrochloride 646 29339990 251579-55-2 (N-acetyl-N-methylglycyl)glycylvalyl-D-alloisoleucylthreonylnorvalylisoleucylarginyl(N-ethylprolinamide) monoacetate (salt) 581 29339990 252742-72-6 5-(chloromethyl)-1,2-dihydro-3H-1,2,4-triazol-3-one 246 29339990 269731-84-2 (5R,6R)-1-benzyl-5-hydroxy-6-(methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one 563 29339990 272107-22-9 3,10-dibromo-8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridine 420 29339990 31560-19-7 N-benzoyl-4-hydroxyproline 421 29339990 31560-20-0 methyl N-benzoyl-4-hydroxyprolinate 91 29339990 32065-66-0 2-(dimethoxymethyl)quinoxaline 1,4-dioxide 741 29339990 346412-97-3 1-aminopyridazinium hexafluorophosphate(1-) 373 29339990 39968-33-7 3H-[1,2,3]triazolo[4,5-b]pyridin-3-ol 645 29339990 442526-89-8 isoleucylarginyl(N-ethylprolinamide) dihydrochloride 729 29339990 481659-93-2 ethyl 1-methyl-5-[4'-(trifluoromethyl)biphenyl-2-carboxamido]indole-2-carboxylate 730 29339990 481659-96-5 potassium 1-methyl-5-[4'-(trifluoromethyl)biphenyl-2-carboxamido]indole-2-carboxylate 311 29339990 5424-01-1 3-aminopyrazine-2-carboxylic acid 724 29339990 61607-68-9 1-[2-(dimethylamino)ethyl]-4,5-dihydro-1H-tetrazole-5-thione 488 29339990 62893-24-7 (6-ethyl-4,5-dioxohexahydropyridazine-3-carboxamido)(4-hydroxyphenyl)acetic acid 223 29339990 6548-09-0 5-bromotryptophan 728 29339990 71056-57-0 ethyl 1-methyl-5-nitroindole-2-carboxylate 19 29339990 75302-98-6 2-tert-butoxy-2-oxoethyl [1-(4-chlorobenzoyl)-5-methoxy-2-methylindol-3-yl]acetate 537 29339990 84946-20-3 2-chloro-1-(4-fluorobenzyl)benzimidazole hydrochloride 72 29339990 86404-63-9 1-(2,4-difluorophenyl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one 396 29339990 92992-17-1 1-(methoxycarbonyl)-2,3-dihydro-1H-pyrrolizine-7-carboxylic acid 416 29339990 96314-26-0 (4S)-4-phenyl-L-proline 737 29341000 115065-79-7 (2E)-2-(2-{[(benzyloxy)carbonyl]amino}-1,3-thiazol-4-yl)-5-[(3-methylbut-2-en-1-yl)oxy]-5-oxopent-2-enoic acid 651 29341000 136401-69-9 (Z)-5-{4-[2-(5-ethylpyridin-2-yl)ethoxy]benzylidene}-1,3-thiazolidine-2,4-dione 643 29341000 161798-03-4 ethyl 2-(3-formyl-4-isobutoxyphenyl)-4-methylthiazole-5-carboxylate 485 29341000 162208-27-7 O-[2-(2-amino-1,3-thiazol-4-yl)-2-((Z)-methoxyimino)acetyl] O, O-diethyl phosphorothioate 725 29341000 162208-28-8 O-(2-(2-aminothiazol-4-yl)-2-{[1-(tert-butoxycarbonyl)-1-methylethoxy]imino}acetyl) O',O''-diethyl phosphorothioate 46 29341000 179258-52-7 tert-butyl (7Z)-7-(2-amino-1,3-thiazol-5-yl)-4-ethoxy-10,10-dimethyl-6-oxo-3,5,9-trioxa-8-aza-4-phosphaundec-7-en-11-oate 4-oxide 247 29341000 186538-00-1 3-[(2S,3S)-2-hydroxy-3-(3-hydroxy-2-methylbenzamido)-4-phenylbutanoyl]-5,5-dimethyl-N-(2-methylbenzyl)-1,3-thiazolidine-4-carboxamide 104 29341000 189448-35-9 (7R)-7-[(2E)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-(hydroxyimino)acetamido]-3-[(3-{[(2-aminoethyl)sulfanyl]methyl}pyridin-4-yl)sulfanyl]-3,4-didehydrocepham-4-carboxylic acid 388 29341000 213252-19-8 5-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]-2-methoxy-N-[4-(trifluoromethyl)benzyl]benzamide 178 29341000 221671-63-2 potassium (2-{N-[4-(4-chloro-2,5-dimethoxyphenyl)-5-(2-cyclohexylethyl)-1,3-thiazol-2-yl]carbamoyl}-5,7-dimethylindolin-1-yl)acetate 111 29341000 224631-15-6 2,5-dioxopyrrolidin-1-yl N-{N-[(2-isopropyl-1,3-thiazol-4-yl)methyl]-N-methylcarbamoyl}-L-valinate 723 29341000 29676-71-9 (2-amino-1,3-thiazol-4-yl)acetic acid 871 29341000 302962-49-8 N-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)thiazole-5-carboxamide or dasatanib (proposed INN) 338 29341000 34272-64-5 (4-methyl-2-sulfanyl-1,3-thiazol-5-yl)acetic acid 859 29341000 478410-84-3 (4R)-N-allyl-3-[(2S,3S)-2-hydroxy-3-(3-hydroxy-2-methylbenzamido)-4-phenylbutanoyl]-5,5-dimethylthiazolidine-4-carboxamide 415 29341000 88023-65-8 potassium 3-[(2-formamido-1,3-thiazol-4-yl)oxoacetamido]-2-methyl-4-oxoazetidine-1-sulfonate 957 29349990 0-00-0 potassium 5-methyl-1,3,4-oxadiazole-2-carboxylate 53 29349990 100988-63-4 1-[((7R)-7-amino-4-carboxy-3,4-didehydrocepham-3-yl)methyl]pyridinium iodide 520 29349990 102212-98-6 N4-benzoyl-2'-deoxy-5'-O-(4,4'-dimethoxytrityl)cytidine 3'-(2-cyanoethyl diisopropylphosphoramidite) 795 29349990 103788-59-6 4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]benzaldehyde 55 29349990 103788-65-4 2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-ol 618 29349990 110483-43-7 2'-bromo-2'-deoxy-5-methyluridine 3',5'-diacetate 451 29349990 113891-01-3 diphenylmethyl (2S,5R)-6,6-dibromo-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate 4-oxide 735 29349990 114341-88-7 3-(2-bromopropanoyl)-4,4-dimethyl-1,3-oxazolidin-2-one 343 29349990 127111-98-2 diphenylmethyl (7R)-7-amino-3-(mesyloxy)-3,4-didehydrocepham-4-carboxylate hydrochloride 439 29349990 130800-76-9 5-(3-chloropropyl)-3-methylisoxazole 260 29349990 134379-77-4 4-amino-5-fluoro-1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]pyrimidin-2(1H)-one 447 29349990 135790-89-5 [(2,2-dimethylpropanoyl)oxy]methyl (7R)-7-[(2Z)-2-(2-{(2S)-2-[(tert-butoxycarbonyl)amino]propanamido}-1,3-thiazol-4-yl)-2-(methoxyimino)acetamido]-3,4-didehydrocepham-4-carboxylate 767 29349990 13636-02-7 (RS)-3-(dimethylamino)-1-(2-thienyl)propan-1-ol 344 29349990 140128-37-6 diphenylmethyl (7R)-7-(2-{2-[(tert-butoxycarbonyl)amino]-1,3-thiazol-4-yl}-2- [(trityloxy)imino]acetamido)-3-({[(1H-1,2,3-triazol-4-yl)sulfanyl]methyl}sulfanyl)-3,4-didehydrocepham-4-carboxylate 177 29349990 155990-20-8 N-[(1-{[2-(diethylamino)ethyl]amino}-7-methoxy-9-oxo-9H-thioxanthen-4-yl)methyl]formamide 8 29349990 158878-46-7 6-{(E)-2-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]vinyl}-4-hydroxytetrahydro-2H-pyran-2-one 771 29349990 164015-32-1 N-methyl-3-(1-naphthyloxy)-2-(2-thienyl)propan-1-amine phosphate 815A 29349990 170985-86-1 1-[(2S,3S)-2-(benzyloxy)pentan-3-yl]-4-(4-{4-[4-({(3R,5R)-5-(2,4-difluorophenyl)-5-[(1H-1,2,4-triazol-1-yl)methyl]tetrahydrofuran-3-yl}methoxy)phenyl]piperazin-1-yl}phenyl)-1H-1,2,4-triazol-5(4H)-one 382 29349990 171482-05-6 (2R,3S)-2-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}-3-(4-fluorophenyl)morpholine hydrochloride 181 29349990 176773-87-8 (3R)-3-(methoxymethyl)-7-(4,4,4-trifluorobutoxy)-3,3a,4,5-tetrahydro[1,3]oxazolo[3,4-a]quinolin-1-one 278A 29349990 177587-08-5 N-{5-[2-((6S)-2-amino-4-oxo-3,4,5,6,7,8-hexahydropyrido[2,3-d]pyrimidin-6-yl)ethyl]-4-methylthiophene-2-carbonyl}-L-glutamic acid 175 29349990 181640-09-5 3-(1-{2-[4-benzoyl-2-(3,4-difluorophenyl)morpholin-2-yl]ethyl}-4-phenylpiperidin-4-yl)-1,1-dimethylurea hydrochloride 125 29349990 182133-09-1 6-(benzyloxy)-3-bromo-2-(4-methoxyphenyl)-1-benzothiophene 1-oxide 659 29349990 183433-66-1 [6-chloro-4-(2-ethyl-1,3-dioxolan-2-yl)-2-methoxypyridin-3-yl]methanol 242 29349990 183434-04-0 tert-butyl (4S)-4-ethyl-4,6-dihydroxy-3,10-dioxo-3,4,8,10-tetrahydro-1H-pyrano[3,4-f]indolizine-7-carboxylate 182 29349990 185835-97-6 (5S)-5-(methoxymethyl)-3-[6-(4,4,4-trifluorobutoxy)-1,2-benzoxazol-3-yl]-1,3-oxazolidin-2-one 185 29349990 186348-69-6 7-chloro-8-[((2R)-1,4-diazabicyclo[2.2.2]octan-2-yl)methylamino]-2,3-dihydro-1,4-benzodioxine-5-carboxamide 656 29349990 18686-82-3 1,3,4-thiadiazole-2-thiol 252 29349990 188016-51-5 methyl N-(butoxycarbonyl)-3-{[(5R)-3-(4-cyanophenyl)-4,5-dihydroisoxazol-5-yl]acetamido}-L-alaninate 187 29349990 189003-92-7 2-{7-fluoro-2-oxo-4-[2-(4-thieno[3,2-c]pyridin-4-ylpiperazin-1-yl)ethyl]quinolin-1(2H)-yl}acetamide 216 29349990 189028-95-3 (4S)-3-[(5R)-5-(4-fluorophenyl)-5-hydroxypentanoyl]-4-phenyl-1,3-oxazolidin-2-one 186 29349990 191023-43-5 5-(8-amino-7-chloro-2,3-dihydro-1,4-benzodioxin-5-yl)-3-(1-phenethylpiperidin-4-yl)-1,3,4-oxadiazol-2(3H)-one 697 29349990 192049-49-3 4-nitrobenzyl 2-((1R,5R)-3-benzyl-7-oxo-4-thia-2,6-diazabicyclo[3.2.0]hept-2-en-6-yl)-3-methylbut-2-enoate 327 29349990 194861-99-9 ((5S)-3-tert-butyl-2-phenyl-1,3-oxazolidin-5-yl)methanol 627 29349990 195708-14-6 (2R,3R,4S)-4-(1,3-benzodioxol-5-yl)-3-(ethoxycarbonyl)-2-(4-methoxyphenyl)pyrrolidinium (2S)-hydroxy(phenyl)acetate 340 29349990 197897-11-3 1-[((7R)-7-amino-4-carboxy-3,4-didehydrocepham-3-yl)methyl]-1H-imidazo[1,2-b]pyridazin-4-ium iodide 30 29349990 199327-61-2 7-methoxy-6-(3-morpholinopropoxy)quinazolin-4(3H)-one 310 29349990 204990-60-3 (3S,10R,13Z,16S)-10-(3-chloro-4-methoxybenzyl)-3-isobutyl-6,6-dimethyl-16-[(1S)-1-((2R,3R)-3-phenyloxiran-2-yl)ethyl]-1,4-dioxa-8,11-diazacyclohexadec-13-ene-2,5,9,12-tetrone 446 29349990 20893-30-5 2-thienylacetonitrile 704B 29349990 220997-99-9 (5R)-9-chloro-5-ethyl-5-hydroxy-10-methyl-12-[(4-methylpiperidin-1-yl)methyl]-1,4,5,13-tetrahydro-3H,15H-oxepino[3',4':6,7]indolizino[1,2-b]quinoline-3,15-dione hydrochloride 704 29349990 221054-70-2 (5R)-5-ethyl-5-hydroxy-1,4,5,8-tetrahydrooxepino[3,4-c]pyridine-3,9-dione 184 29349990 223570-85-2 8-methyl-8-azabicyclo[3.2.1]octan-3-yl 2,3-dihydropyrazolo[1,5,4-de][1,4]benzoxazine-6-carboxylate 432 29349990 223595-20-8 (1R)-5-(1,3,6,2-dioxazaborocan-2-yl)-1-methyl-2-tritylisoindoline 707 29349990 227029-27-8 2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl methanesulfonate 299 29349990 227625-35-6 3-{[2-(aminomethyl)cyclohexyl]methyl}-1,2,4-oxadiazol-5(4H)-one 298 29349990 227626-65-5 tert-butyl N-methyl-N-{2-[(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)methyl]cyclohexyl}carbamate 299A 29349990 227626-75-7 3-{[2-(aminomethyl)cyclohexyl]methyl}-1,2,4-oxadiazol-5(4H)-one hydrochloride 300 29349990 229336-92-9 3-chloro-N-{4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl}-4-{[2-(methylamino)imidazol-1-yl]methyl}thiophene-2-carboxamide 300A 29349990 229340-73-2 3-chloro-N-{4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl}-4-{[2-(methylamino)imidazol-1-yl]methyl}thiophene-2-carboxamide trifluoroacetate 722 29349990 24209-43-6 (7R)-7-amino-3-[2-(1,3,4-thiadiazol-2-ylsulfanyl)ethyl]-3,4-didehydrocepham-4-carboxylic acid 82 29349990 252317-48-9 {(3S)-1-[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl]pyrrolidin-3-yl}diphenylacetonitrile 289 29349990 253450-09-8 6-({2-[4-(4-fluorobenzyl)piperidin-1-yl]ethyl}sulfinyl)-1,3-benzoxazol-2(3H)-one 841 29349990 253450-12-3 6-{[2-(4-benzylpiperidin-1-yl)ethyl]sulfinyl}-1,3-benzoxazol-2(3H)-one 408 29349990 287737-72-8 (2S)-hydroxy(phenyl)acetic acid — (1S)-3-(dimethylamino)-1-(2-thienyl)propan-1-ol (1:1) (salt) 383 29349990 287930-73-8 4-benzyl-2-hydroxymorpholin-3-one 384 29349990 287930-75-0 (2R)-4-benzyl-2-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}morpholin-3-one 325 29349990 30165-96-9 4-(4-chloro-1,2,5-thiadiazol-3-yl)morpholine 815 29349990 345217-03-0 2-[(2S,3S)-2-(benzyloxy)pentan-3-yl]-4-(4-{4-[4-({(3R,5R)-5-(2,4-difluorophenyl)-5-[(1H-1,2,4-triazol-1-yl)methyl]tetrahydrofuran-3-yl}methoxy)phenyl]piperazin-1-yl}phenyl)semicarbazide 854 29349990 362543-73-5 DNA, d(P-thio) (C-T-A-G-A-T-T-T-C-C-C-G-C-G), tridecasodium salt 448 29349990 36923-17-8 (7R)-7-amino-3,4-didehydrocepham-4-carboxylic acid 717 29349990 37539-03-0 (7R)-7-amino-3-[(1H-1,2,3-triazol-4-ylsulfanyl)methyl]-3,4-didehydrocepham-4-carboxylic acid 832 29349990 377727-87-2 2-(2-furyl)-7-(2-{4-[4-(2-methoxyethoxy)phenyl]piperazin-1-yl}ethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[2,3-c]pyrimidin-5-amine 706B 29349990 475479-34-6 (2S)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]-1-benzothiophen-7-yl}propanoic acid 706 29349990 475480-88-7 4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]-1-benzothiophene-7-carbaldehyde 959 29349990 518048-05-0 potassium 4-[N-(2-fluorobenzyl)carbamoyl]-1-methyl-2-[1-methyl-1-(5-methyl-1,3,4-oxadiazole-2-carboxamido)ethyl]-6-oxo-1,6-dihydropyrimidine-5-olate 707A 29349990 521266-46-6 (2S)-1-{N-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl]glycyl}pyrrolidine-2-carbonitrile 655 29349990 53994-69-7 (7R)-7-amino-3-chloro-3,4-didehydrocepham-4-carboxylic acid 719 29349990 61807-78-1 7-(bromoacetamido)-7-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)lsulfanyl]methyl}-3,4-didehydrocepham-4-carboxylic acid 738 29349990 63457-21-6 diphenylmethyl 2-(3-benzyl-7-oxo-4-thia-2,6-diazabicyclo[3.2.0]hept-2-en-6-yl)-3-methylbut-3-enoate 961 29349990 635724-55-9 (2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine succinate 797 29349990 649761-25-1 methyl N-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]benzyl}glycinate hydrochloride 702 29349990 655233-39-9 4-nitrobenzyl (7R)-7-amino-3-((2S)-tetrahydrofuran-2-yl)-3,4-didehydrocepham-4-carboxylate hydrochloride 769 29349990 663603-70-1 (2Z)-3-(methylamino)-1-(2-thienyl)prop-2-en-1-one 721 29349990 68350-02-7 (7R)-7-amino-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-3,4-didehydrocepham-4-carboxylic acid hydrochloride 718 29349990 70035-75-5 diphenylmethyl (7S)-7-(bromoacetamido)-7-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-3,4-didehydrocepham-4-carboxylate 855 29349990 744239-10-9 DNA, d(P-thio) (G-A-T-C-C-G-C-G-G-G-A-A-A-T), tridecasodium salt 665 29349990 7481-90-5 1-(3,5-anhydro-2-deoxy-β-D-threo-pentofuranosyl)-5-methylpyrimidine-2,4(1H,3H)-dione 208 29349990 75776-79-3 1,4-dithia-7-azaspiro[4.4]nonane-8-carboxylic acid hydrobromide 93 29349990 76646-91-8 (3S)-6,6-dibromo-2,2-dimethylpenam-3-carboxylic acid 1,1-dioxide 90 29349990 76801-85-9 (2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-13-[(2,6-dideoxy-3-C-methyl-3-O-methyl-α-L-ribo-hexopyranosyl)oxy]-2-ethyl-3,4,10-trihydroxy-3,5,8,10,12,14-hexamethyl-11-{[3,4,6-trideoxy-3-(dimethylamino)-β-D-xylo-hexopyranosyl]oxy}-1-oxa-6-azacyclopentadecan-15-one 716 29349990 79349-82-9 trans-(7R)-7-amino-3-vinyl-3,4-didehydrocepham-4-carboxylic acid 243 29349990 86639-52-3 (4S)-4,11-diethyl-4,9-dihydroxy-1H,12H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione 952 29349990 872728-82-0 N-[4-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)phenyl]glycine 342 29349990 92096-37-2 diphenylmethyl (7R)-3-(mesyloxy)-7-(phenylacetamido)-3,4-didehydrocepham-4-carboxylate 525 29349990 93183-15-4 2'-deoxy-5'-O-(4,4'-dimethoxytrityl)-N2-isobutyrylguanosine 3'-(2-cyanoethyl diisopropylphosphoramidite) 688 29349990 96219-87-3 (3-aminopyrazol-4-yl)(2-thienyl)methanone 584 29349990 98-03-3 thiophene-2-carbaldehyde 526 29349990 98796-51-1 2'-deoxy-5'-O-(4,4'-dimethoxytrityl)thymidine 3'-(2-cyanoethyl diisopropylphosphoramidite) 527 29349990 98796-53-3 N6-benzoyl-2'-deoxy-5'-O-(4,4'-dimethoxytrityl)adenosine 3'-(2-cyanoethyl diisopropylphosphoramidite) 517 29349990 98819-76-2 (2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine 770 29349990 116539-55-0 (1S)-3-(methylamino)-1-(2-thienyl)propan-1-ol 179 29350090 137431-02-8 N-[3-(2-amino-1-hydroxyethyl)-4-fluorophenyl]methanesulfonamide 626a 29350090 141430-65-1 N-[2-(4-hydroxyanilino)pyridin-3-yl]-4-methoxybenzene-1-sulfonamide 329 29350090 149490-60-8 N-(butane-1-sulfonyl)-L-tyrosine 328 29350090 149490-61-9 N-(butane-1-sulfonyl)-O-(4-pyridin-4-ylbutyl)-L-tyrosine 40 29350090 160231-69-6 (3S)-tetrahydrofuran-3-yl N-[(2S,3R)-3-hydroxy-4-(N-isobutyl-4-nitrobenzene-1-sulfonamido)-1-phenylbutan-2-yl]carbamate 562 29350090 169280-56-2 4-amino-N-[(2R,3S)-3-amino-2-hydroxy-4-phenylbutyl]-N-isobutylbenzene-1-sulfonamide 711 29350090 170569-88-7 4-[5-(4-fluorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzene-1-sulfonamide 691 29350090 186497-07-4 N-(3-methoxy-5-methylpyrazin-2-yl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-3-sulfonamide 180 29350090 189814-01-5 3-(2-amino-1-hydroxyethyl)-4-methoxybenzene-1-sulfonamide 88 29350090 200575-15-1 4-[2-ethoxy-5-(4-methylpiperazine-1-sulfonyl)benzamido]-1-methyl-3-propylpyrazole-5-carboxamide 587 29350090 210538-75-3 N-(1,2,3,4-tetrahydroisoquinolin-5-yl)methanesulfonamide hydrochloride 41 29350090 244634-31-9 N-((2R,3S)-3-amino-2-hydroxy-4-phenylbutyl)-N-isobutyl-4-nitrobenzene-1-sulfonamide hydrochloride 75 29350090 247582-73-6 2-ethoxy-5-(4-ethylpiperazine-1-sulfonyl]nicotinic acid 224 29350090 289042-12-2 (4R,6S)-6-((E)-2-{4-(4-fluorophenyl)-6-isopropyl-2-[mesyl(methyl)amino]pyrimidin-5-yl}vinyl)-2,2-dimethyl-1,3-dioxan-4-yl 3,3-dimethylbutanoate 592 29350090 334826-98-1 5-[2-ethoxy-5-(4-ethylpiperazine-1-sulfonyl)pyridin-3-yl]-3-ethyl-2-(2-methoxyethyl)-2,3,4,5,6,7-hexahydropyrazolo[4,3-d]pyrimidin-7-one 593 29350090 334827-99-5 5-[2-ethoxy-5-(4-ethylpiperazine-1-sulfonyl)pyridin-3-yl]-3-ethyl-2-(2-methoxyethyl)-2,3,4,5,6,7-hexahydropyrazolo[4,3-d]pyrimidin-7-one 4-methylbenzene-1-sulfonate 591 29350090 334828-19-2 N-[3-carbamoyl-5-ethyl-1-(2-methoxyethyl)pyrazol-4-yl]-2-ethoxy-5-[(4-ethylpiperazin-1-yl)sulfonyl]nicotinamide 596 29350090 364321-71-1 3-[(dimethylamino)methyl]-4-[4-(methylsulfanyl)phenoxy]benzene-1-sulfonamide 597 29350090 364323-49-9 3-[(dimethylamino)methyl]-4-[4-(methylsulfanyl)phenoxy]benzene-1-sulfonamide L-tartarate (1:1) 70 29350090 88933-16-8 1-(4-hydrazinophenyl)-N-methylmethanesulfonamide hydrochloride 335 29389090 517-43-1 mixture of sennoside A and B 336 29389090 52730-36-6, 52730-37-7 mixture of sennoside A and B, calcium salts 882 29391900 58-00-4 (6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de, g]quinoline-10,11-diol or apomorphine 666 29392000 467430-13-3 2-[2-methyl-1-(propionyloxy)propoxy]-2-[(4-phenylbutyl)phosphinoyl]acetic acid, (9R)-cinchonan-9-ol salt (1:1) 617 29400000 270071-40-4 benzyl 2,6-dimethoxy-4-{(5R,5aR,8aR,9S)-6-oxo-9-[(2,3,4,6-tetra-O-benzyl-β-D-glucopyranosyl)oxy]-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol-5-yl}phenyl carbonate 667 29400000 471863-88-4 2,3-di-O-benzyl-4,6-O-((1R)-ethylidene)-D-xylo-hexopyranose 668 29400000 473799-30-3 (5S,5aS,9S)-9-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxo-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol-5-yl 2,3-di-O-benzyl-4,6-O-[(1R)-ethylidene]-β-D-glucopyranoside 616 29400000 6564-72-3 2,3,4,6-tetra-O-benzyl-D-glucopyranose 15 29419000 19130-96-2 (2S,3S,4R,5R)-2-(hydroxymethyl)piperidine-3,4,5-triol 200 29419000 54122-50-8 dicyclohexylammmonium (7R)-3-(acetoxymethyl)-7-[2-({(3R)-3-[(tert-butoxycarbonyl)amino]-3-carboxypropyl}amino)-2-oxoethyl]-3,4-didehydrocepham-4-carboxylate or cephalosporin D dicyclohexylamine salt 131 30021095 42617-41-4 Blood-coagulation factor XIVa 321 38249098 127852-28-2 (1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethan-1-ol, acetonitrile solution 510 38249098 170277-77-7 (3S)-3-[2-(mesyloxy)ethoxy]-4-(trityloxy)butyl methanesulfonate, dimethylformamide solution 326 38249098 30165-96-9 4-(4-chloro-1,2,5-thiadiazol-3-yl)morpholine, toluene solution 409 38249098 38345-66-3 (2S,3R)-4-(dimethylamino)-3-methyl-1,2-diphenylbutan-2-ol, toluene solution 132 38249098 84449-81-0 4-[2-(piperidin-1-yl)ethoxy]benzoyl chloride hydrochloride, 1,2-dichloroethane solution

ANNEX IV List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be withdrawn from the list of products receiving duty-free treatment included in Annex 6 to Regulation (EC) No 1549/2006

ID No CN code CAS RN Name 677 29189090 157283-68-6 isopropyl (Z)-7-[(1R,2R,3R,5S)-3,5-dihydroxy-2-{(E)-(3R)-3-hydroxy-4-[3-(trifluoromethyl)phenoxy]but-1-enyl}cyclopentyl]hept-5-enoate travoprost (INN) 603 29242995 112522-64-2 4-acetamido-2'-aminobenzanilide tacedinaline (INN) 69 29242995 166518-60-1 N-[(2,6-diisopropylphenoxy)sulfonyl]-2-(2,4,6-triisopropylphenyl)acetamide avasimibe (INN) 441 29280090 53016-31-2 13-ethyl-17-alpha-hydroxy-18,19-dinorpregn-4-en-20-yn-3-one oxime norelgestromin (INN) 833 29309030 583-91-5 2-hydroxy-4-(methylthio)butyric acid desmeninol (INN) 273 29329970 114870-03-0 methyl O-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranosyl-(1,4)-O-beta-D-glucopyranuronosyl-(1,4)-O-2-deoxy-3,6-di-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranosyl-(1,4)-O-2-O-sulfo-alpha-L-idopyranuronosyl-(1,4)-2-deoxy-2-(sulfoamino)-6-(hydrogen sulfate)-alpha-D-glucopyranoside, decasodium salt fondaparinux sodium (INN) 627 29333999 75970-99-9 [1-(4-fluorobenzyl)-1H-benzimidazol-2-yl](4-piperidyl)amine tecastemizole (INN) 159 29333999 100643-71-8 8-chloro-11-(4-piperidylidene)-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridine desloratadine (INN) 549 29333999 168273-06-1 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidino-1H-pyrazole-3-carboxamide rimonabant (INN) 380 29333999 193275-84-2 4-{4-[(11R)-3,10-dibromo-8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl]piperidinocarbonylmethyl}piperidine-1-carboxamide lonafarnib (INN) 397 29334990 146362-70-1 2-{[1-(7-chloro-4-quinolyl)-5-(2,6-dimethoxyphenyl)-1H-pyrazol-3-yl]carbonylamino}adamantane-2-carboxylic acid meclinertant (INN) 641 29335995 147127-20-6 (R)-[2-(6-amino-9H-purin-9-yl)-1-methylethoxy]methylphosphonic acid tenofovir (INN) 205 29335995 149950-60-7 6-benzyl-1-(ethoxymethyl)-5-isopropylpyrimidine-2,4(1H,3H)-dione emivirine (INN) 511 29335995 153537-73-6 (S)-2-(4-{[(2,7-dimethyl-4-oxo-1,4-dihydroquinazolin-6-yl)methyl](prop-2-ynyl)amino}-2-fluorobenzamido)-4-(1H-tetrazol-5-yl)butyric acid plevitrexed (INN) 686 29349990 112984-60-8 (+-)-6-fluoro-1-methyl-4-oxo-7-(piperazin-1-yl)-4H-[1,3]thiazeto[3,2-a]quinoline-3-carboxylic acid ulifloxacin (INN) 33 29349990 145514-04-1 (2R,4R)-4-(2,6-diamino-9H-purin-9-yl)-1,3-dioxolan-2-ylmethanol amdoxovir (INN) 513 29349990 171228-49-2 4-[4-(4-{4-[(3R,5R)-5-(2,4-difluorophenyl)-5-(1H-1,2,4-triazol-1-ylmethyl)tetrahydrofuran-3-ylmethyloxy]phenyl}piperazin-1-yl)phenyl]-1-[(1S,2S)-1-ethyl-2-hydroxypropyl]-1,2,4-triazol-5(4H)-one posaconazole (INN) 293 29349990 184475-35-2 (3-chloro-4-fluorophenyl)[7-methoxy-6-(3-morpholinopropoxy)quinazolin-4-yl]amine gefitinib (INN) 539 29350090 150375-75-0 N'-{(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-3-hydroxy-2,3-dihydro-1H-indol-2-ylcarbonyl}-L-prolinamide relcovaptan (INN) 39 29350090 161814-49-9 (3S)-tetrahydrofuran-3-yl (1S,2R)-3-[(4-aminophenylsulfonyl)(isobutyl)amino]-1-benzyl-2-hydroxypropylcarbamate amprenavir (INN) 115 29350090 169590-42-5 4-[5-(p-tolyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide celecoxib (INN) 654 29350090 180200-68-4 4-(4-cyclohexyl-2-methyloxazol-5-yl)-2-fluorobenzenesulfonamide tilmacoxib (INN) 690 29350090 181695-72-7 4-(5-methyl-3-phenylisoxazol-4-yl)benzenesulfonamide valdecoxib (INN) 520 29350090 192329-42-3 (S)-N-hydroxy-2,2-dimethyl-4-[4-(4-pyridyloxy)phenylsulfonyl]-1,4-thiazinane-3-carboxamide prinomastat (INN) 364 30021095 193700-51-5 SC-70935 leridistim (INN)

Versions

1. 2007-02-12